SCHEMBL21190843

SCHEMBL21190843

CC1(C)OB(c2cc(CS(C)(=O)=O)ccc2Nc2ccc(F)cc2F)OC1(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 7/20 0.45
ALDH1A1 P00352 1/20 0.36
PTGS2 P35354 1/20 0.36
GSK3A P49840 1/20 0.36
CDK9 P50750 1/20 0.36
IRAK1 P51617 1/20 0.36
SOS1 Q07889 1/20 0.36
GAA P10253 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
BRD2 P25440 1/20 0.34
BRD3 Q15059 1/20 0.34
BRDT Q58F21 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
PKM P14618 1/20 0.34
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
KDR P35968 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155173 0.90 BRD4 (0.36) BRD4ALDH1A1PTGS2SOS1GAA
SCHEMBL21190844 0.88 BRD4 (0.44) BRD4PTGS2SOS1CA1CA2
SCHEMBL15069481 0.81 BRD4 (0.48) BRD4PTGS2GSK3ACDK9IRAK1
SCHEMBL21190847 0.81 BRD4 (0.42) BRD4ALDH1A1PTGS2CDK9GAA
SCHEMBL20155117 0.80 ALDH1A1 (0.39) ALDH1A1PTGS2SOS1GAACA1
SCHEMBL21190848 0.79 BRD4 (0.44) BRD4PTGS2GAACA1CA2
SCHEMBL9937303 0.78 LPL (0.36) GSK3ACDK9IRAK1CA1CA2
SCHEMBL20155541 0.76 ALDH1A1 (0.40) ALDH1A1PTGS2SOS1GAACA1
SCHEMBL16009256 0.76 BRD4 (0.51) BRD4ALDH1A1PTGS2GSK3ACDK9
SCHEMBL20157282 0.75 LIPG (0.37) BRD4CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200354371-A1 BROMODOMAIN INHIBITOR COMPOUND AND USE THEREOF SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2020-11-12 US disclosed
WO-2019141131-A1 BROMODOMAIN INHIBITOR COMPOUND AND USE THEREOF 中国科学院上海药物研究所 2019-07-25 WO disclosed
US-9359548-B2 Organic electroluminescent device UDC IRELAND LIMITED (IE) 2016-06-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200354371-A1 BROMODOMAIN INHIBITOR COMPOUND AND USE THEREOF BRD4, BRD1, BRD3 BRD4 1/4885ALDH1A1 3333/4885PTGS2 3990/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.