SCHEMBL20155541

SCHEMBL20155541

CC1(C)OB(c2cc(N)c(F)cc2Nc2ccc(F)cc2F)OC1(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
LPL P06858 1/20 0.36
LIPG Q9Y5X9 1/20 0.36
SOS1 Q07889 1/20 0.35
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
GAA P10253 2/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
NFKB1 P19838 1/20 0.32
RAB9A P51151 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HTT P42858 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
HDAC1 Q13547 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155498 0.89 ALDH1A1 (0.36) ALDH1A1LPLLIPGSOS1CYP2D6
SCHEMBL20155117 0.86 ALDH1A1 (0.39) ALDH1A1LPLLIPGSOS1CYP2D6
SCHEMBL20155588 0.79 ALDH1A1 (0.37) ALDH1A1LPLLIPGSOS1CYP2D6
SCHEMBL21190843 0.76 BRD4 (0.45) ALDH1A1SOS1CA1CA2CA9
SCHEMBL20155120 0.74 ALDH1A1 (0.40) ALDH1A1LPLLIPGPTGS2
SCHEMBL20155461 0.74 TDO2 (0.38) ALDH1A1LPLLIPGCA1CA2
SCHEMBL15289502 0.74 LPL (0.37) ALDH1A1LPLLIPG
SCHEMBL29395754 0.74 LPL (0.49) ALDH1A1LPLLIPGCA1CA2
SCHEMBL772615 0.74 LPL (0.49) ALDH1A1LPLLIPGCA1CA2
SCHEMBL20155620 0.73 EGFR (0.37) CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed