SCHEMBL20156083

SCHEMBL20156083

CCOC(=O)C[C@H](NC(=O)/C(=C/NCc1cc2c(nc1C)NCCC2)C(=N)COC(C)(C)C)c1ccc(OC)c(F)c1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 16/20 0.40
ITGAV P06756 16/20 0.40
ITGB6 P18564 6/20 0.37
ITGA2B P08514 1/20 0.37
ITGB5 P18084 6/20 0.37
ITGB8 P26012 5/20 0.37
PDE2A O00408 2/20 0.32
MAPK1 P28482 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20156349 0.87 ITGB3 (0.49) ITGB3ITGAVITGB6ITGA2BITGB5
SCHEMBL20156078 0.85 RXFP1 (0.35) PDE2AMEN1ALDH1A1KMT2A
SCHEMBL20156283 0.84 ITGB3 (0.38) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL20156301 0.80 ITGB3 (0.57) ITGB3ITGAVITGB6ITGA2BITGB5
SCHEMBL23912904 0.78 ITGAV (0.39) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL21281625 0.78 ITGB3 (0.40) ITGB3ITGAVITGB6ITGA2BITGB5
SCHEMBL23912908 0.77 NPC1 (0.34) ITGB3ITGAVPDE2AMAPK1MEN1
SCHEMBL23912902 0.73 ITGB3 (0.53) ITGB3ITGAVITGB6ITGA2BITGB5
SCHEMBL23912864 0.71 ITGB3 (0.60) ITGB3ITGAVITGB6ITGA2BITGB5
SCHEMBL20156082 0.71 ITGB3 (0.49) ITGB3ITGAVITGB6ITGA2BITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538527-B1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2021-10-13 EP disclosed
WO-2018089358-A1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed