SCHEMBL20156349

SCHEMBL20156349

CCOC(=O)C[C@H](NC(=O)/C(=C/NCCc1ccc2c(n1)NCCC2)C(=N)COC(C)(C)C)c1ccc(OC)c(F)c1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 19/20 0.49
ITGAV P06756 19/20 0.49
ITGB6 P18564 13/20 0.46
ITGB5 P18084 13/20 0.46
ITGB8 P26012 12/20 0.46
ITGA2B P08514 1/20 0.46
CXCR4 P61073 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20156301 0.93 ITGB3 (0.57) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL20156083 0.87 ITGB3 (0.40) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL23912902 0.86 ITGB3 (0.53) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL23912908 0.85 NPC1 (0.34) ITGB3ITGAV
SCHEMBL23912864 0.84 ITGB3 (0.60) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL20156034 0.84 ITGAV (0.49) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL20156291 0.84 ITGB3 (0.62) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL20156282 0.81 ITGB3 (0.57) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL20156250 0.80 ITGAV (0.52) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL20156082 0.79 ITGB3 (0.49) ITGB3ITGAVITGB6ITGB5ITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538527-B1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2021-10-13 EP disclosed
WO-2018089358-A1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed