SCHEMBL20156944

SCHEMBL20156944

C[C@H](N)CNc1cc(F)c(C#N)cc1F

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 2/20 0.40
ADRB2 P07550 2/20 0.38
ADRB1 P08588 2/20 0.38
BACE2 Q9Y5Z0 1/20 0.33
KHK P50053 1/20 0.32
USP30 Q70CQ3 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
ADRB3 P13945 1/20 0.31
CYP2D6 P10635 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
NOS2 P35228 1/20 0.30
CYP11B1 P15538 2/20 0.30
CYP11B2 P19099 2/20 0.30
TRPV3 Q8NET8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20156962 0.77 TRPV4 (0.44) TRPV4ADRB2ADRB1BACE2KHK
SCHEMBL3628472 0.72 TRPV4 (0.50) TRPV4ADRB2ADRB1BACE2KHK
SCHEMBL3186092 0.72 TRPV4 (0.50) TRPV4ADRB2ADRB1BACE2KHK
SCHEMBL14566112 0.70 PKM (0.42)
SCHEMBL6651303 0.69 TRPV4 (0.71) TRPV4KHKCYP11B1CYP11B2
SCHEMBL4624565 0.66 TRPV4 (0.43) TRPV4USP30
SCHEMBL2081398 0.65 TRPV4 (0.45) TRPV4ADRB2ADRB1BACE2KHK
SCHEMBL12413852 0.65 TRPV4 (0.50) TRPV4ADRB2ADRB1KHKCYP11B1
SCHEMBL366972 0.64 TRPV4 (0.65) TRPV4KHKCYP11B1CYP11B2
SCHEMBL26106182 0.64 ACLY (0.36) TRPV4ADRB2ADRB1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed