SCHEMBL20156962

SCHEMBL20156962

N#Cc1cc(F)c(NCCN)cc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 2/20 0.44
FERMT2 Q96AC1 1/20 0.36
KHK P50053 1/20 0.35
USP30 Q70CQ3 1/20 0.34
BACE2 Q9Y5Z0 1/20 0.33
ALDH1A1 P00352 2/20 0.33
CHEK1 O14757 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
CA12 O43570 1/20 0.33
CA3 P07451 1/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33
CA5A P35218 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
CA5B Q9Y2D0 1/20 0.33
DPP4 P27487 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3628472 0.77 TRPV4 (0.50) TRPV4KHKUSP30BACE2ADRB2
SCHEMBL20156944 0.77 TRPV4 (0.40) TRPV4KHKUSP30BACE2ADRB2
SCHEMBL21180029 0.74 KAT2B (0.49) FERMT2USP30ALDH1A1KDM4EKAT2B
SCHEMBL3186092 0.73 TRPV4 (0.50) TRPV4KHKUSP30BACE2ADRB2
SCHEMBL6651303 0.73 TRPV4 (0.71) TRPV4KHKALDH1A1CYP11B1CYP11B2
SCHEMBL24056640 0.72 CHEK1 (0.49) FERMT2CHEK1
SCHEMBL21704265 0.71 ALDH1A1 (0.47) ALDH1A1KDM4EHSD17B10
SCHEMBL26106182 0.71 ACLY (0.36) TRPV4BACE2ADRB2ADRB1
SCHEMBL30317451 0.70 TSHR (0.58) FERMT2ALDH1A1KDM4ECA12CA3
SCHEMBL20156858 0.70 TSHR (0.58) FERMT2ALDH1A1KDM4ECA12CA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed