SCHEMBL20157094

SCHEMBL20157094

C=C(CCCC)c1ccc(N)c(C(=C)C)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B3 P37058 1/20 0.33
HTR7 P34969 1/20 0.33
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
SKP2 Q13309 1/20 0.33
ALDH1A1 P00352 2/20 0.32
HSD17B10 Q99714 2/20 0.32
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32
NOS2 P35228 2/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
MAPT P10636 1/20 0.31
STS P08842 1/20 0.31
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
CYP1A2 P05177 2/20 0.30
TSHR P16473 2/20 0.30
LMNA P02545 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11696345 0.74 LMNA (0.47) HSD17B3HTR7ESR1ESR2ALDH1A1
SCHEMBL10270183 0.73 TSHR (0.44) ALDH1A1HSD17B10MAPTKDM4ECYP1A2
SCHEMBL24633879 0.73 PDE4A (0.37) HSD17B3ESR1ESR2ALDH1A1HSD17B10
SCHEMBL23865855 0.72 KDM4E (0.39) HTR7ALDH1A1HSD17B10THRBMAPT
SCHEMBL5496843 0.72 ERAP2 (0.49) ALDH1A1HSD17B10HDAC1MAPTKDM4E
SCHEMBL28930606 0.70 HSD17B3 (0.37) HSD17B3HTR7ESR1ESR2ALDH1A1
SCHEMBL2017777 0.70 TSHR (0.49) ALDH1A1HDAC1HDAC8TSHRSLC6A2
SCHEMBL20686672 0.69 ESR1 (0.49) HSD17B3ESR1ESR2ALDH1A1CYP1A2
SCHEMBL7193415 0.69 ALDH1A1 (0.44) HSD17B3HTR7ESR1ESR2ALDH1A1
SCHEMBL7187984 0.69 HSD17B3 (0.60) HSD17B3ESR1ESR2ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed