SCHEMBL20157701

SCHEMBL20157701

Cc1ccc(C(O)c2cc(Cl)c(C)cc2Br)cc1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.39
S1PR1 P21453 1/20 0.35
BRD4 O60885 2/20 0.33
SLC6A2 P23975 6/20 0.32
SLC6A4 P31645 6/20 0.32
SLC6A3 Q01959 6/20 0.32
CYP3A4 P08684 5/20 0.31
CYP2D6 P10635 5/20 0.31
CYP2C19 P33261 1/20 0.31
MLKL Q8NB16 1/20 0.31
MAPK1 P28482 1/20 0.31
S1PR4 O95977 1/20 0.31
S1PR3 Q99500 1/20 0.31
KCNH2 Q12809 4/20 0.31
THRB P10828 1/20 0.31
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157702 0.88 ATM (0.40) LMNAS1PR1BRD4SLC6A2SLC6A4
SCHEMBL21362758 0.80 S1PR3 (0.38) S1PR1BRD4MAPK1S1PR3
SCHEMBL20157931 0.78 GAA (0.38) LMNASLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL21362626 0.78 ALDH1A1 (0.31) LMNACYP3A4CYP2D6CYP2C19MLKL
SCHEMBL20157428 0.78 MLKL (0.35) LMNABRD4SLC6A2CYP3A4CYP2D6
SCHEMBL20157996 0.73
SCHEMBL16169582 0.71 ALDH1A1 (0.41) LMNABRD4CYP3A4CYP2C19MLKL
SCHEMBL15958523 0.71 LMNA (0.59) LMNAS1PR1CYP3A4MAPK1
SCHEMBL20157371 0.71 ACHE (0.44) LMNABRD4MEN1MAPTKMT2A
SCHEMBL21352143 0.71 BRD4 (0.34) BRD4THRBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed