SCHEMBL21362626

SCHEMBL21362626

CCc1cc(C(O)c2ccc(C)cc2)c(Br)cc1C

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.31
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ACHE P22303 1/20 0.31
CYP3A4 P08684 2/20 0.31
CYP2D6 P10635 2/20 0.31
CYP2C19 P33261 2/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
KMT2A Q03164 1/20 0.31
MAPT P10636 1/20 0.31
IGF1R P08069 1/20 0.30
THRA P10827 1/20 0.30
THRB P10828 1/20 0.30
MLKL Q8NB16 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157701 0.78 LMNA (0.39) LMNACYP3A4CYP2D6CYP2C19MEN1
SCHEMBL20157931 0.76 GAA (0.38) LMNASMN1; SMN2ACHECYP3A4CYP2C19
SCHEMBL20157428 0.75 MLKL (0.35) ALDH1A1LMNAACHECYP3A4CYP2D6
SCHEMBL21362510 0.71 OPRK1 (0.38) ALDH1A1SMN1; SMN2
SCHEMBL21362758 0.71 S1PR3 (0.38)
SCHEMBL20157996 0.71
SCHEMBL16169582 0.69 ALDH1A1 (0.41) ALDH1A1LMNACYP3A4CYP2C19MEN1
SCHEMBL21352143 0.69 BRD4 (0.34) KMT2ATHRATHRB
SCHEMBL20157371 0.69 ACHE (0.44) ALDH1A1LMNAACHEMEN1KMT2A
SCHEMBL11854000 0.68 MLKL (0.41) ALDH1A1LMNACYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed