SCHEMBL20159006

SCHEMBL20159006

Cn1cc(CN2CCC(Nc3ccccc3Cl)CC2)cc1C(=O)N1CCN(c2ccc(F)cc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 5/20 0.47
PTGS1 P23219 1/20 0.45
PTGS2 P35354 1/20 0.45
TP53 P04637 1/20 0.45
PRKAA2 P54646 3/20 0.44
KMT2A Q03164 1/20 0.44
HRH3 Q9Y5N1 2/20 0.43
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
SIGMAR1 Q99720 2/20 0.41
SLC6A12 P48065 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
MCHR1 Q99705 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159115 0.85 MTOR (0.55) PTGS1PTGS2HRH3
SCHEMBL20159010 0.81 PTGS1 (0.45) PTGS1PTGS2TP53KDM4E
SCHEMBL20159008 0.81 NPY2R (0.51) PTGS1PTGS2HRH3
SCHEMBL20159066 0.79 MTOR (0.45) PTGS1PTGS2HRH3
SCHEMBL20159024 0.78 MTOR (0.64) KMT2AHRH3
SCHEMBL20159009 0.77 PTGS1 (0.46) PTGS1PTGS2TP53HRH3
SCHEMBL20159286 0.77 MTOR (0.51) HRH3
SCHEMBL20159079 0.76 MTOR (0.52) CHRM4HRH3
SCHEMBL20159109 0.73 MTOR (0.50) CHRM4PTGS1PTGS2TP53
SCHEMBL20139225 0.73 MTOR (0.50) CHRM4KMT2AHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed