SCHEMBL20159009

SCHEMBL20159009

Cn1cc(CN2CCC3(CCN(c4ccccc4Cl)C3)C2)cc1C(=O)N1CCN(c2ccc(F)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.46
PTGS2 P35354 1/20 0.46
CYP2D6 P10635 8/20 0.43
CYP3A4 P08684 4/20 0.43
CYP1A2 P05177 3/20 0.43
MTOR P42345 1/20 0.43
RPTOR Q8N122 1/20 0.43
MLST8 Q9BVC4 1/20 0.43
TSHR P16473 4/20 0.42
POLB P06746 1/20 0.42
CYP2C19 P33261 2/20 0.41
HPGD P15428 1/20 0.41
USP2 O75604 2/20 0.41
CYP2C9 P11712 2/20 0.41
TP53 P04637 1/20 0.41
HRH3 Q9Y5N1 1/20 0.40
AR P10275 1/20 0.40
HIF1A Q16665 1/20 0.40
RECQL P46063 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159115 0.87 MTOR (0.55) PTGS1PTGS2MTORRPTORMLST8
SCHEMBL20159066 0.81 MTOR (0.45) PTGS1PTGS2MTORRPTORMLST8
SCHEMBL20159286 0.81 MTOR (0.51) MTORRPTORMLST8POLBHRH3
SCHEMBL20159024 0.80 MTOR (0.64) MTORRPTORMLST8POLBHRH3
SCHEMBL20159008 0.79 NPY2R (0.51) PTGS1PTGS2MTORRPTORMLST8
SCHEMBL20159079 0.78 MTOR (0.52) MTORRPTORMLST8POLBHRH3
SCHEMBL20159006 0.77 CHRM4 (0.47) PTGS1PTGS2TP53HRH3
SCHEMBL20159010 0.76 PTGS1 (0.45) PTGS1PTGS2MTORRPTORMLST8
Trifluoroacetic Acid SCHEMBL20139757 0.75 MTOR (0.50) MTORRPTORMLST8POLBHRH3
SCHEMBL20159109 0.75 MTOR (0.50) PTGS1PTGS2MTORRPTORMLST8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed