SCHEMBL20159910

SCHEMBL20159910

CCOC(=O)Nc1cc(-c2cc(N)ccc2Oc2ccc(F)cc2F)nn2cnnc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
BRD4 O60885 13/20 0.38
BRPF1 P55201 1/20 0.38
KCNQ3 O43525 3/20 0.37
KCNQ2 O43526 3/20 0.37
KCNQ4 P56696 1/20 0.37
KCNQ5 Q9NR82 1/20 0.37
LMNA P02545 1/20 0.35
ABCB11 O95342 1/20 0.35
ESR1 P03372 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA2A P08913 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
ALOX15 P16050 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159922 0.87 BRD4 (0.47) BRD4
SCHEMBL20159918 0.86 BRPF1 (0.53) NPC1MAPTRAB9ABRD4BRPF1
SCHEMBL20160087 0.78 BRD4 (0.40) NPC1MAPTRAB9ABRD4BRPF1
SCHEMBL20160243 0.76 BRPF1 (0.51) NPC1MAPTRAB9ABRD4BRPF1
SCHEMBL20159916 0.75 BRD9 (0.41) MAPTBRD4BRPF1
SCHEMBL20159867 0.75 BRD9 (0.56) MAPTBRD4BRPF1
SCHEMBL20160293 0.72 BRD4 (0.43) NPC1BRD4LMNA
SCHEMBL20160050 0.70 BRD4 (0.46) BRD4BRPF1
SCHEMBL20160415 0.70 ALDH1A1 (0.46) MAPTBRD4BRPF1CYP1A2CYP2C9
SCHEMBL20160251 0.69 BRD4 (0.41) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed