SCHEMBL20159984

SCHEMBL20159984

Nc1ccc(Oc2ccc(F)cc2P)c(-c2ccc3nncn3n2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.35
BRD4 O60885 2/20 0.34
NPC1 O15118 1/20 0.34
HTT P42858 1/20 0.34
GAA P10253 1/20 0.33
KDM4E B2RXH2 4/20 0.33
PSMD14 O00487 1/20 0.33
USP2 O75604 1/20 0.33
PRNP P04156 1/20 0.33
POLB P06746 1/20 0.33
MMP2 P08253 1/20 0.33
PTPN7 P35236 1/20 0.33
PPARG P37231 1/20 0.33
RECQL P46063 1/20 0.33
PPP1CA P62136 1/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
PTPN22 Q9Y2R2 1/20 0.33
NR2E3 Q9Y5X4 1/20 0.33
NCOR2 Q9Y618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20160293 0.89 BRD4 (0.43) SMN1; SMN2BRD4NPC1HTTGAA
SCHEMBL20160417 0.71 BRD4 (0.42) SMN1; SMN2BRD4NPC1HTTKDM4E
SCHEMBL20160024 0.69 BRD4 (0.45) SMN1; SMN2BRD4KDM4EKMT2ATDP1
SCHEMBL20159904 0.67 MAPK14 (0.41) BRD4
SCHEMBL20160308 0.67 BRD4 (0.43) BRD4KMT2A
SCHEMBL20159910 0.65 NPC1 (0.39) BRD4NPC1LMNAMAPT
SCHEMBL11629082 0.65 KDM4E (0.53) SMN1; SMN2GAAKDM4EPOLBPPARG
SCHEMBL10389609 0.64 ALDH1A1 (0.50) SMN1; SMN2HTTGAAKDM4EPOLB
SCHEMBL11628077 0.63 KDM4E (0.46) SMN1; SMN2NPC1HTTGAAKDM4E
SCHEMBL20160255 0.62 ATM (0.40) BRD4KMT2ATDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed