SCHEMBL20161606

SCHEMBL20161606

CCNc1cc(OC)nc(N)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.44
NPC1 O15118 2/20 0.44
ALDH1A1 P00352 2/20 0.44
TLR8 Q9NR97 2/20 0.42
AURKA O14965 1/20 0.42
PDPK1 O15530 1/20 0.42
TGFBR1 P36897 1/20 0.42
AURKB Q96GD4 1/20 0.42
NUDT1 P36639 4/20 0.41
PGK1 P00558 2/20 0.40
GRM4 Q14833 1/20 0.40
KCNH2 Q12809 1/20 0.39
CACNA1C Q13936 1/20 0.39
SCN5A Q14524 1/20 0.39
ADORA3 P0DMS8 2/20 0.38
ADORA1 P30542 1/20 0.38
MAPK1 P28482 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
ADORA2A P29274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20434304 0.83 TLR8 (0.65) RAB9ANPC1ALDH1A1TLR8MAPK1
SCHEMBL8873492 0.80 PGK1 (0.40) RAB9ANPC1ALDH1A1TLR8AURKA
SCHEMBL8347788 0.80 NPC1 (0.47) RAB9ANPC1ALDH1A1PGK1KCNH2
SCHEMBL16463778 0.79 NUDT1 (0.60) RAB9ANPC1ALDH1A1NUDT1GRM4
SCHEMBL8873249 0.78 TLR8 (0.37) RAB9ANPC1ALDH1A1TLR8AURKA
SCHEMBL10102121 0.77 TLR8 (0.47) RAB9ANPC1TLR8AURKAPDPK1
SCHEMBL151590 0.76 ALDH1A1 (0.59) RAB9ANPC1ALDH1A1AURKAPDPK1
SCHEMBL18177432 0.76 DHFR (0.53) NPC1ALDH1A1MAPK1
SCHEMBL8630748 0.76 NPC1 (0.56) RAB9ANPC1ALDH1A1AURKAPDPK1
SCHEMBL6128303 0.76 TLR8 (0.69) RAB9ANPC1TLR8AURKAPDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018087602-A1 RESOLUTION OF OPTICALLY ACTIVE DIAZASPIRO[4.5]DECANE DERIVATIVES ROIVANT SCIENCES GMBH (CH) 2018-05-17 WO disclosed