Cgp-12177

Cgp-12177

SCHEMBL2016211

CC(C)(C)NCC(O)COc1cccc2[nH]c(=O)[nH]c12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 8/20 1.00
ADRB1 P08588 5/20 1.00
ADRB3 P13945 5/20 1.00
CYP1A2 P05177 3/20 1.00
MEN1 O00255 2/20 1.00
KMT2A Q03164 2/20 1.00
ALOX15 P16050 1/20 1.00
LMNA P02545 1/20 0.98
CYP2D6 P10635 3/20 0.70
SLC6A4 P31645 2/20 0.70
SLC6A2 P23975 1/20 0.70
CASR P41180 1/20 0.70
SLC6A3 Q01959 1/20 0.70
KCNH2 Q12809 1/20 0.70
KDM4E B2RXH2 2/20 0.57
ALDH1A1 P00352 2/20 0.57
MAPT P10636 2/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2C19 P33261 1/20 0.57
TDP1 Q9NUW8 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cgp-12177 SCHEMBL12329633 1.00 ADRB2 (1.00) ADRB2ADRB1ADRB3CYP1A2MEN1
Cgp-12177 SCHEMBL4538049 0.99 ADRB2 (1.00) ADRB2ADRB1ADRB3CYP1A2MEN1
SCHEMBL10594616 0.89 ADRB3 (0.80) ADRB2ADRB1ADRB3CYP1A2MEN1
SCHEMBL11230530 0.86 ADRB2 (0.76) ADRB2ADRB1ADRB3CYP1A2MEN1
SCHEMBL11331685 0.86 ADRB2 (0.75) ADRB2ADRB1ADRB3CYP1A2MEN1
Hydrochloric Acid SCHEMBL11462740 0.85 ADRB2 (0.76) ADRB2ADRB1ADRB3CYP1A2MEN1
SCHEMBL11242745 0.84 ADRB2 (0.73) ADRB2ADRB1ADRB3CYP1A2MEN1
Hydrochloric Acid SCHEMBL11248041 0.83 ADRB2 (0.73) ADRB2ADRB1ADRB3CYP1A2MEN1
SCHEMBL16187027 0.83 ADRB2 (0.71) ADRB2ADRB1ADRB3CYP1A2MEN1
SCHEMBL16189744 0.83 ADRB2 (0.71) ADRB2ADRB1ADRB3CYP1A2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 222 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250360149-A1 GPCR INHIBITORS AND USES THEREOF GPCR THERAPEUTICS INC (KR) 2025-11-27 US claimed
EP-4536239-A1 GPCR INHIBITORS AND USES THEREOF GPCR Therapeutics, Inc. (KR) 2025-04-16 EP claimed
WO-2025050038-A2 GPCR INHIBITORS AND USES THEREOF GPCR THERAPEUTICS, INC. (KR) 2025-03-06 WO claimed
CN-119562815-A GPCR inhibitors and uses thereof GPCR治疗公司 2025-03-04 CN claimed
US-20240301022-A1 GLYCOPROTEINS HAVING LIPID MOBILIZING PROPERTIES AND THERAPEUTIC USES THEREOF UNIV ASTON (GB) 2024-09-12 US claimed
WO-2023239937-A1 GPCR INHIBITORS AND USES THEREOF GPCR THERAPEUTICS, INC. (KR) 2023-12-14 WO claimed
WO-2022198259-A1 TREATMENT METHODS FOR PULMONARY ARTERIAL HYPERTENSION THE HEART RESEARCH INSTITUTE LTD (AU) 2022-09-29 WO claimed
US-20220273751-A1 GPCR HETEROMER INHIBITORS AND USES THEREOF GPCR THERAPEUTICS, INC. (KR) 2022-09-01 US claimed
EP-3969007-A1 GPCR HETEROMER INHIBITORS AND USES THEREOF GPCR Therapeutics, Inc. (KR) 2022-03-23 EP claimed
CN-114051416-A GPCR heteromer inhibitors and uses thereof GPCR治疗公司 2022-02-15 CN claimed
CN-114028370-A Composition with effects of preventing and treating obesity and related diseases and application thereof 中山大学 2022-02-11 CN claimed
EP-4199925-B1 CYCLOPENTAPYRROLE OREXIN RECEPTOR AGONISTS MERCK SHARP & DOHME LLC (US) 2026-05-20 EP disclosed
EP-3558298-B1 ANTIDIABETIC SPIROCHROMAN COMPOUNDS MERCK SHARP & DOHME LLC (US) 2026-03-11 EP disclosed
US-12552767-B2 3-heteroaryl pyrrolidine and piperidine orexin receptor agonists MERCK SHARP & DOHME LLC (US) 2026-02-17 US disclosed
US-20260021061-A1 ARIADNE AND ANALOGS FOR THE TREATMENT OF NEUROLOGICAL AND NEUROMUSCLAR DISORDERS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2026-01-22 US disclosed
WO-2004089288-A2 METHOD OF TREATING LOWER URINARY TRACT DISORDERS DYNOGEN PHARMACEUTICALS, INC. (US) 2004-10-21 WO disclosed
US-20040198822-A1 Methods for treating lower urinary tract disorders using alpha2delta subunit calcium channel modulators with smooth muscle modulators DYNOGEN PHARMACUETICALS, INC. (US) 2004-10-07 US disclosed
WO-2004066990-A2 METHODS OF TREATING LOWER URINARY TRACT DISORDERS USING SODIUM CHANNEL MODULATORS DYNOGEN PHARMACEUTICALS, INC. (US) 2004-08-12 WO disclosed
EP-0003298-B1 4-HYDROXY-2-BENZIMIDAZOLIN-THION DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM Roche Diagnostics GmbH (DE) 1981-03-25 EP disclosed
EP-0000784-A1 4-Hydroxy-2-benzimidazolinone derivatives, process for their preparation and their use in medicaments Roche Diagnostics GmbH (DE) 1979-02-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040198822-A1 Methods for treating lower urinary tract disorders using alpha2delta subunit calcium channel modulators with smooth muscle modulators GABRB2, GABRD, GABRB3 ADRB2 19/4885ADRB1 60/4885ADRB3 71/4885
US-12552767-B2 3-heteroaryl pyrrolidine and piperidine orexin receptor agonists HCRTR2, HCRTR1, NPY1R ADRB2 177/4885ADRB1 161/4885ADRB3 131/4885
US-20260021061-A1 ARIADNE AND ANALOGS FOR THE TREATMENT OF NEUROLOGICAL AND NEUROMUSCLAR DISORDERS ATXN2, HCRTR2, CDR2 ADRB2 135/4885ADRB1 487/4885ADRB3 120/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.