SCHEMBL20162423

SCHEMBL20162423

CC(C)(C)C1(c2ccccc2-c2cncn2C2CC2)CCCN1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.42
MARK3 P27448 1/20 0.42
MAP4K2 Q12851 1/20 0.42
CAMK2B Q13554 1/20 0.42
PIM3 Q86V86 1/20 0.42
PIM2 Q9P1W9 1/20 0.42
HSP90AA1 P07900 2/20 0.38
HSP90AB1 P08238 2/20 0.38
TDO2 P48775 8/20 0.38
IDO1 P14902 16/20 0.37
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20162427 0.77 CYP11B1 (0.36) HSP90AA1HSP90AB1IDO1CYP3A4
SCHEMBL3312128 0.71 NPSR1 (0.35)
SCHEMBL3313722 0.71 NPSR1 (0.35)
SCHEMBL3312135 0.71 NPSR1 (0.35)
SCHEMBL20162418 0.68 IDO1 (0.48) TDO2IDO1CYP3A4
SCHEMBL16730871 0.65 PIM1 (0.55) PIM1MARK3MAP4K2CAMK2BPIM3
SCHEMBL17007540 0.65 LMNA (0.40)
SCHEMBL20164006 0.64 ALDH1A1 (0.43)
SCHEMBL20164004 0.64 ALDH1A1 (0.43)
SCHEMBL29150660 0.64 CD44 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068391-B1 ARYL LINKED IMIDAZOLE AND TRIAZOLE DERIVATIVES AND METHODS OF USE THEREOF FOR IMPROVING THE PHARMACOKINETICS OF A DRUG MERCK SHARP & DOHME (US) 2018-05-23 EP claimed