SCHEMBL2016541

SCHEMBL2016541

O=C(N[C@H]1C[C@@H]1c1ccccc1)C1CCC(c2ccccc2)N(S(=O)(=O)c2ccccc2)C1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
RAB9A P51151 1/20 0.52
KMT2A Q03164 1/20 0.52
EPHX2 P34913 2/20 0.49
TLR2 O60603 12/20 0.47
TLR1 Q15399 11/20 0.47
SMN1; SMN2 Q16637 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
KDM1A O60341 1/20 0.44
TGM2 P21980 1/20 0.43
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12628187 0.85 ALDH1A1 (0.53) ALDH1A1RAB9AKMT2AEPHX2GAA
SCHEMBL2018212 0.85 ALDH1A1 (0.53) ALDH1A1RAB9AKMT2AEPHX2GAA
SCHEMBL2016241 0.82 ALDH1A1 (0.52) ALDH1A1RAB9AKMT2AEPHX2GAA
SCHEMBL2016436 0.82 ALDH1A1 (0.52) ALDH1A1RAB9AKMT2AEPHX2GAA
SCHEMBL12628299 0.82 ALDH1A1 (0.52) ALDH1A1RAB9AKMT2AEPHX2GAA
SCHEMBL12629087 0.81 ALDH1A1 (0.65) ALDH1A1RAB9AKMT2ASMN1; SMN2
SCHEMBL2011747 0.81 ALDH1A1 (0.65) ALDH1A1RAB9AKMT2ASMN1; SMN2
SCHEMBL12628172 0.81 ALDH1A1 (0.57) ALDH1A1RAB9AKMT2AEPHX2
SCHEMBL2013828 0.81 ALDH1A1 (0.57) ALDH1A1RAB9AKMT2ASMN1; SMN2GAA
SCHEMBL12629075 0.81 ALDH1A1 (0.57) ALDH1A1RAB9AKMT2ASMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073269-A1 PIPERIDINE ARYL SULFONAMIDE DERIVATIVES AS KV1.3 MODULATORS EVOTEC AG (DE) 2011-06-23 WO claimed