SCHEMBL20170692

SCHEMBL20170692

CN[C@H]1Cc2ccc(OC)c3c2C2[C@@H](NCC[C@@H]21)O3

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.36
MRGPRX2 Q96LB1 1/20 0.31
MAPT P10636 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
HTR2C P28335 1/20 0.30
ACHE P22303 1/20 0.30
ADRA1A P35348 2/20 0.30
HTR1A P08908 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13072367 0.74 OPRM1 (0.34) HCRTR1
SCHEMBL20170650 0.73 HCRTR1 (0.44) HCRTR1ADRA1AHTR1A
SCHEMBL20170778 0.70 HCRTR1 (0.33) HCRTR1
SCHEMBL13972294 0.66 HCRTR1 (0.41) HCRTR1MRGPRX2HTR1A
SCHEMBL18473438 0.66 HCRTR1 (0.41) HCRTR1MRGPRX2HTR1A
SCHEMBL13972295 0.66 HCRTR1 (0.41) HCRTR1MRGPRX2HTR1A
SCHEMBL20170731 0.64 HCRTR1 (0.43) HCRTR1HTR1A
SCHEMBL20170703 0.64 HCRTR1 (0.47) HCRTR1MRGPRX2MAPTHTR1A
SCHEMBL20170880 0.64 HCRTR1 (0.45) HCRTR1HTR1A
SCHEMBL20170657 0.63 MTNR1A (0.43) HCRTR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2453895-B1 (+) - MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF MALLINCKRODT LLC (US) 2018-05-23 EP disclosed