SCHEMBL20172295

SCHEMBL20172295

CCCCCOc1cc(N)ncn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.41
MCHR1 Q99705 3/20 0.40
TLR8 Q9NR97 3/20 0.40
SOAT1 P35610 1/20 0.38
SMPD1 P17405 1/20 0.37
CDK1 P06493 2/20 0.36
CCNB1 P14635 2/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CCNA1 P78396 1/20 0.36
ADORA2A P29274 1/20 0.35
GABRP O00591 2/20 0.35
GABRD O14764 2/20 0.35
GABRA1 P14867 2/20 0.35
GABRB1 P18505 2/20 0.35
GABRG2 P18507 2/20 0.35
GABRB3 P28472 2/20 0.35
GABRA5 P31644 2/20 0.35
GABRA3 P34903 2/20 0.35
GABRA2 P47869 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16291043 0.89 MAPT (0.38) MCHR1TLR8GABRPGABRDGABRA1
SCHEMBL720347 0.86 SOAT1 (0.42) TSHRTLR8SOAT1SMPD1GABRP
SCHEMBL10188104 0.80 ALDH1A1 (0.39) TSHRTLR8GABRPGABRDGABRA1
SCHEMBL31548577 0.80 GABRP (0.44) TSHRTLR8SOAT1GABRPGABRD
SCHEMBL11373823 0.79 PIK3CD (0.37) TSHR
SCHEMBL15933181 0.77 CA2 (0.39)
SCHEMBL2237291 0.76 HTR7 (0.46)
SCHEMBL10187279 0.76 MCHR1 (0.41) MCHR1
SCHEMBL15114929 0.73 LMNA (0.44) TSHRSOAT1GABRPGABRDGABRA1
SCHEMBL18578440 0.73 MCHR1 (0.56) TSHRMCHR1TLR8SOAT1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3323414-A1 INHIBITORS OF NEDD8-ACTIVATING ENZYME Millennium Pharmaceuticals, Inc. (US) 2018-05-23 EP disclosed