SCHEMBL20177860

SCHEMBL20177860

O=C(N[C@@H]1c2nncn2C[C@H]1c1c(F)cc(Br)cc1F)OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 2/20 0.48
KDM1A O60341 2/20 0.39
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSK P43235 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
DPP4 P27487 4/20 0.36
DPP7 Q9UHL4 4/20 0.36
HSD11B1 P28845 1/20 0.35
KCNH2 Q12809 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177491 0.89 CCKBR (0.47) CCKBRCTSLCTSBCTSK
SCHEMBL20177635 0.86 KDM1A (0.41) CCKBRKDM1ACTSLCTSBCTSK
SCHEMBL20177518 0.77 CCKBR (0.41) CCKBRCTSLCTSBCTSKALDH1A1
SCHEMBL20177567 0.76 FPR2 (0.52) CTSL
SCHEMBL20177674 0.76 KDM1A (0.42) CCKBRKDM1ACTSLALDH1A1GAA
SCHEMBL18270477 0.75 FPR2 (0.45) CCKBR
SCHEMBL20177919 0.75 KDM1A (0.41) CCKBRKDM1ACTSLALDH1A1GAA
SCHEMBL22068860 0.73 CA1 (0.44) CCKBRCTSLCTSBCTSK
SCHEMBL20177845 0.73 BRD4 (0.47) CTSLCTSBCTSK
SCHEMBL20177499 0.73 SMN1; SMN2 (0.37) ALDH1A1GAAKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed