SCHEMBL20179716

SCHEMBL20179716

CCCCCCC[C@H]1CC[C@H](CC(=O)N(CCC)[C@@H](CC(C)C2=C(C)[C@@H](C)[C@H](c3ccccc3)O2)C(=O)NCc2cccs2)CC1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPR88 Q9GZN0 1/20 0.34
F12 P00748 5/20 0.33
ALOX5 P09917 3/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
HPGD P15428 1/20 0.32
ALDH1A1 P00352 3/20 0.32
GAA P10253 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
MAPK1 P28482 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30
TSHR P16473 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20179720 0.91 GPR88 (0.35) GPR88F12ALOX5KMT2AHPGD
SCHEMBL20179718 0.82 F12 (0.31) F12ALDH1A1SMN1; SMN2
SCHEMBL20179719 0.81 F12 (0.37) F12KMT2AMEN1HPGDALDH1A1
SCHEMBL20179717 0.74 TSHR (0.40) ALOX5HPGDALDH1A1GAANPSR1
SCHEMBL20179646 0.66 GAA (0.43) GPR88KMT2AMEN1HPGDALDH1A1
SCHEMBL20179645 0.62 GPR88 (0.41) GPR88ALOX5KMT2AMEN1HPGD
SCHEMBL20179555 0.61 HPGD (0.62) GPR88KMT2AMEN1HPGDALDH1A1
SCHEMBL20179732 0.61 USP2 (0.45) KMT2AMEN1HPGDALDH1A1GAA
SCHEMBL27753473 0.58 GAA (0.41) KMT2AMEN1HPGDALDH1A1GAA
SCHEMBL27733090 0.58 GAA (0.41) KMT2AMEN1HPGDALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018093695-A1 FACTOR XIIa INHIBITORS MERCK SHARP & DOHME CORP. (US) 2018-05-24 WO disclosed