SCHEMBL20179718

SCHEMBL20179718

CCCN(C(=O)CC1CCC(N=[N+]=[N-])CC1)[C@@H](CC(C)C1=C(C)[C@@H](C)[C@H](c2ccccc2)O1)C(=S)NCc1cccs1

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
F12 P00748 2/20 0.31
ALDH1A1 P00352 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20179720 0.84 GPR88 (0.35) F12ALDH1A1SMN1; SMN2
SCHEMBL20179716 0.82 GPR88 (0.34) F12ALDH1A1SMN1; SMN2
SCHEMBL20179645 0.73 GPR88 (0.41) ALDH1A1SMN1; SMN2
SCHEMBL20179717 0.68 TSHR (0.40) ALDH1A1SMN1; SMN2
SCHEMBL20179646 0.60 GAA (0.43) ALDH1A1SMN1; SMN2
SCHEMBL21571092 0.57 F12 (0.71) F12
SCHEMBL21579639 0.57 F12 (0.65) F12
SCHEMBL21571084 0.57 F12 (0.71) F12
SCHEMBL6076695 0.55 KMT2A (0.66) ALDH1A1
SCHEMBL28195196 0.54 HSD11B1 (0.54) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018093695-A1 FACTOR XIIa INHIBITORS MERCK SHARP & DOHME CORP. (US) 2018-05-24 WO disclosed