SCHEMBL20179720

SCHEMBL20179720

CCCN(C(=O)C[C@H]1CC[C@H](N)CC1)[C@@H](CC(C)C1=C(C)[C@@H](C)[C@H](c2ccccc2)O1)C(=O)NCc1cccs1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPR88 Q9GZN0 1/20 0.35
F12 P00748 4/20 0.34
ALOX5 P09917 3/20 0.33
ALDH1A1 P00352 3/20 0.33
GAA P10253 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MAPK1 P28482 1/20 0.32
TSHR P16473 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
POLB P06746 2/20 0.31
KMT2A Q03164 1/20 0.31
HTT P42858 2/20 0.31
USP2 O75604 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20179716 0.91 GPR88 (0.34) GPR88F12ALOX5ALDH1A1GAA
SCHEMBL20179718 0.84 F12 (0.31) F12ALDH1A1SMN1; SMN2
SCHEMBL20179646 0.76 GAA (0.43) GPR88ALDH1A1GAANPSR1TSHR
SCHEMBL20179717 0.76 TSHR (0.40) ALOX5ALDH1A1GAANPSR1TSHR
SCHEMBL20179645 0.63 GPR88 (0.41) GPR88ALOX5ALDH1A1GAANPSR1
SCHEMBL20179732 0.59 USP2 (0.45) ALDH1A1GAANPSR1TSHRSMN1; SMN2
SCHEMBL20179555 0.59 HPGD (0.62) GPR88ALDH1A1GAANPSR1TSHR
SCHEMBL6076695 0.59 KMT2A (0.66) ALDH1A1GAATSHRPOLBKMT2A
SCHEMBL20363266 0.58 GAA (0.63) ALDH1A1GAANPSR1TSHRSMN1; SMN2
SCHEMBL17712437 0.57 GAA (0.61) ALDH1A1GAANPSR1TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018093695-A1 FACTOR XIIa INHIBITORS MERCK SHARP & DOHME CORP. (US) 2018-05-24 WO disclosed