SCHEMBL20180449

SCHEMBL20180449

COc1cc(I)ccc1N1CCNCC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 8/20 0.61
HTR3E A5X5Y0 3/20 0.61
HTR3B O95264 3/20 0.61
HTR3A P46098 3/20 0.61
HTR3D Q70Z44 3/20 0.61
HTR3C Q8WXA8 3/20 0.61
DRD2 P14416 2/20 0.61
DRD3 P35462 2/20 0.61
ADRB1 P08588 2/20 0.61
CYP2C19 P33261 1/20 0.61
SIGMAR1 Q99720 1/20 0.61
LMNA P02545 1/20 0.59
MAPT P10636 1/20 0.59
HTR7 P34969 3/20 0.51
HTR1A P08908 1/20 0.51
HTR1D P28221 1/20 0.51
HTR1B P28222 1/20 0.51
HTR2C P28335 1/20 0.51
ADRA1B P35368 1/20 0.51
HTR2B P41595 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24518342 0.82 DRD2 (0.60) HTR6DRD2DRD3MAPTHTR7
SCHEMBL233151 0.82 HTR3A (0.71) HTR6HTR3EHTR3BHTR3AHTR3D
SCHEMBL6709128 0.82 HTR3A (0.63) HTR6HTR3EHTR3BHTR3AHTR3D
SCHEMBL30747759 0.82 HTR3A (0.71) HTR6HTR3EHTR3BHTR3AHTR3D
SCHEMBL30952473 0.81 HTR3A (0.66) HTR6HTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL4905371 0.81 HTR3A (0.69) HTR6HTR3EHTR3BHTR3AHTR3D
SCHEMBL4190135 0.81 HTR6 (0.61) HTR6HTR3EHTR3BHTR3AHTR3D
SCHEMBL31651894 0.81 HTR3E (0.77) HTR6HTR3EHTR3BHTR3AHTR3D
SCHEMBL8874392 0.81 HTR3A (0.61) HTR6HTR3EHTR3BHTR3AHTR3D
SCHEMBL2875715 0.81 HTR3A (0.66) HTR6HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018090939-A1 8,9-DIHYDROIMIDAZOLE[1,2-A]PYRIMIDO[5,4-E]PYRIMIDINE-5(6H)-KETONE COMPOUND 上海瑛派药业有限公司 2018-05-24 WO disclosed