SCHEMBL2018094

SCHEMBL2018094

NCCc1cc(F)c2cccnc2c1N1CCN(C2CCC2)CC1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 14/20 0.43
KDM4E B2RXH2 2/20 0.38
RAD52 P43351 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HRH1 P35367 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
ALDH1A1 P00352 2/20 0.36
LMNA P02545 2/20 0.36
GLA P06280 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ACHE P22303 1/20 0.35
ADRA2A P08913 1/20 0.35
DRD4 P21917 1/20 0.35
HTR2A P28223 1/20 0.35
HTT P42858 1/20 0.34
HIF1A Q16665 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2015675 0.88 METAP2 (0.43) HTR1AKDM4ERAD52L3MBTL1HRH1
SCHEMBL2013524 0.85 HTR1A (0.42) HTR1AKDM4ERAD52L3MBTL1HRH1
SCHEMBL2017390 0.85 METAP2 (0.44) HTR1AKDM4ERAD52L3MBTL1HRH1
SCHEMBL2012338 0.84 KDM4E (0.42) HTR1AKDM4ERAD52L3MBTL1HRH3
SCHEMBL2051072 0.81 HTR1A (0.35) HTR1AKDM4ERAD52L3MBTL1HRH1
SCHEMBL2164993 0.80 HTR1A (0.44) HTR1AKDM4EL3MBTL1HRH1HRH3
SCHEMBL2014289 0.80 KDM4E (0.36) HTR1AKDM4EL3MBTL1ALDH1A1LMNA
SCHEMBL2014290 0.80 KDM4E (0.36) HTR1AKDM4EL3MBTL1ALDH1A1LMNA
SCHEMBL2163161 0.78 HTR1A (0.44) HTR1AKDM4ERAD52L3MBTL1HRH3
SCHEMBL2019128 0.75 METAP2 (0.44) HTR1AKDM4EL3MBTL1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed