SCHEMBL2018189

SCHEMBL2018189

CCn1c(CN)nc2cc(-c3ccc(OC)cc3)ccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.53
MAPT P10636 4/20 0.51
NPC1 O15118 3/20 0.51
RAB9A P51151 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C19 P33261 1/20 0.51
NLRP3 Q96P20 1/20 0.49
PPARG P37231 1/20 0.47
RPS6KA5 O75582 1/20 0.46
GRIK1 P39086 2/20 0.44
GRIK2 Q13002 2/20 0.44
NTRK1 P04629 2/20 0.44
CSF1R P07333 2/20 0.44
NTRK2 Q16620 2/20 0.44
AAK1 Q2M2I8 1/20 0.43
LMNA P02545 3/20 0.42
ALDH1A1 P00352 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2018222 0.90 MAPT (0.51) TDP1MAPTNPC1RAB9ACYP1A2
SCHEMBL2020859 0.87 TDP1 (0.53) TDP1MAPTNPC1RAB9ACYP1A2
SCHEMBL16406373 0.81 ACSS2 (0.53) TDP1MAPTNPC1RAB9ACYP1A2
SCHEMBL21540396 0.77 TDP1 (0.70) TDP1MAPTNPC1RAB9ACYP1A2
SCHEMBL2043847 0.77 PPARG (0.48) TDP1MAPTNPC1RAB9ACYP1A2
SCHEMBL2015354 0.76 PPARG (0.52) TDP1MAPTNPC1RAB9ACYP1A2
SCHEMBL12636234 0.76 MAPT (0.47) TDP1MAPTNPC1RAB9ACYP1A2
SCHEMBL2016798 0.75 KDM4E (0.44) TDP1MAPTNPC1RAB9ACYP1A2
SCHEMBL2017353 0.74 MAPT (0.52) TDP1MAPTNPC1RAB9ACYP1A2
SCHEMBL9195588 0.73 NLRP3 (0.55) RAB9ANLRP3PPARGAAK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed