SCHEMBL2018304

SCHEMBL2018304

CCn1c(CNC(=O)c2nc(Cl)c(N)nc2N)nc2ccc(CCC(=O)OC)cc21

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.40
SCNN1A P37088 9/20 0.39
ACSS2 Q9NR19 3/20 0.37
TSHR P16473 2/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
THPO P40225 1/20 0.36
HSD17B10 Q99714 1/20 0.36
KDM4E B2RXH2 1/20 0.35
GMNN O75496 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
GLA P06280 1/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
PMP22 Q01453 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2014255 0.91 HTT (0.41) HTTSCNN1AACSS2TSHRTP53
SCHEMBL2016749 0.90 ACSS2 (0.41) HTTSCNN1AACSS2TSHRTP53
SCHEMBL12636338 0.88 SCNN1A (0.40) HTTSCNN1AACSS2TSHRTP53
SCHEMBL2018137 0.87 ACSS2 (0.39) HTTSCNN1AACSS2TSHRTP53
SCHEMBL2020338 0.87 HTT (0.46) HTTSCNN1AACSS2TSHRTP53
SCHEMBL2013943 0.86 ACSS2 (0.38) HTTSCNN1AACSS2KMT2A
SCHEMBL2015353 0.86 HTT (0.38) HTTSCNN1AACSS2TSHRTP53
SCHEMBL2018438 0.85 SCNN1A (0.44) HTTSCNN1AACSS2TP53
SCHEMBL2014371 0.85 FKBP1A (0.41) HTTSCNN1AACSS2TSHRTP53
SCHEMBL2015541 0.84 HTT (0.46) HTTACSS2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed