SCHEMBL2014371

SCHEMBL2014371

CCn1c(CNC(=O)c2nc(Cl)c(N)nc2N)nc2ccc(CCC(=O)N3CCOCC3)cc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 3/20 0.41
TSHR P16473 2/20 0.37
HTT P42858 1/20 0.36
ALDH1A1 P00352 3/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
THPO P40225 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PIK3CD O00329 2/20 0.34
MAPK1 P28482 2/20 0.34
KMT2A Q03164 2/20 0.34
LMNA P02545 2/20 0.34
KDM4E B2RXH2 1/20 0.34
GMNN O75496 1/20 0.34
GLA P06280 1/20 0.34
HPGD P15428 1/20 0.34
PMP22 Q01453 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2014255 0.86 HTT (0.41) TSHRHTTALDH1A1TP53CYP1A2
SCHEMBL2018304 0.85 HTT (0.40) TSHRHTTALDH1A1TP53CYP1A2
SCHEMBL2016749 0.85 ACSS2 (0.41) TSHRHTTALDH1A1TP53CYP1A2
Iodide SCHEMBL2015385 0.84 SCNN1A (0.39) FKBP1ATSHRALDH1A1NPSR1TP53
SCHEMBL2018137 0.83 ACSS2 (0.39) TSHRHTTTP53CYP1A2CYP3A4
SCHEMBL2020338 0.83 HTT (0.46) TSHRHTTALDH1A1TP53CYP1A2
SCHEMBL2013943 0.81 ACSS2 (0.38) HTTKMT2AACSS2SCNN1A
SCHEMBL2040435 0.80 HTT (0.45) TSHRHTTALDH1A1TP53CYP1A2
SCHEMBL16882399 0.80 MAPT (0.37) TSHRHTTPIK3CDACSS2
SCHEMBL17937169 0.79 PTGES (0.38) HTTALDH1A1PIK3CDKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed