SCHEMBL20183788

SCHEMBL20183788

CCn1c(=O)cc(C(C)C)c2cc(C(=O)N(C)c3ccc(C(F)(F)F)cc3)ccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.38
KDM4E B2RXH2 1/20 0.38
F2 P00734 1/20 0.38
MCHR1 Q99705 2/20 0.37
MLNR O43193 1/20 0.37
POLQ O75417 1/20 0.37
MLYCD O95822 1/20 0.36
HDAC4 P56524 1/20 0.36
PGR P06401 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NR1H3 Q13133 2/20 0.35
NR1H2 P55055 1/20 0.35
RORC P51449 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
RXRA P19793 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20183836 0.90 MEN1 (0.44) LMNAKDM4EF2POLQPDE4A
SCHEMBL20354318 0.88 KDM4E (0.42) KDM4EF2SMN1; SMN2RORCTP53
SCHEMBL20183659 0.88 RXRA (0.37) LMNAKDM4EPGRRORCTP53
SCHEMBL20183650 0.87 ALDH1A1 (0.41) LMNAKDM4ESMN1; SMN2RORCTP53
SCHEMBL20183824 0.87 RXRA (0.37) KDM4ERORCTP53MAPTRXRA
SCHEMBL20183596 0.87 HDAC8 (0.41) KDM4EMCHR1PGRRORCTP53
SCHEMBL20183791 0.85 ALDH1A1 (0.38) KDM4EF2SMN1; SMN2RORCTP53
SCHEMBL20354281 0.85 KDM4E (0.38) LMNAKDM4ESMN1; SMN2RORCTP53
SCHEMBL20183714 0.84 TUBB4A (0.44) KDM4ERORCTP53MAPT
SCHEMBL21474026 0.83 MAPT (0.41) KDM4EF2SMN1; SMN2RORCTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10987349-B2 Antitumor agent and bromodomain inhibitor FUJIFILM CORPORATION (JP) 2021-04-27 US disclosed
US-10987349-B2 Antitumor agent and bromodomain inhibitor FUJIFILM CORPORATION (JP) 2021-04-27 US disclosed
EP-3563851-B1 ANTITUMOR AGENT AND BROMODOMAIN INHIBITOR FUJIFILM CORP (JP) 2021-04-21 EP disclosed
EP-3327004-B1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND FUJIFILM CORP (JP) 2020-11-04 EP disclosed
US-10696637-B2 Nitrogen-containing heterocyclic compound FUJIFILM CORPORATION (JP) 2020-06-30 US disclosed
US-10696637-B2 Nitrogen-containing heterocyclic compound FUJIFILM CORPORATION (JP) 2020-06-30 US disclosed
US-10633343-B2 2020-04-28 US disclosed
US-10633343-B2 2020-04-28 US disclosed
EP-3563851-A1 ANTITUMOR AGENT AND BROMODOMAIN INHIBITOR FUJIFILM Corporation (JP) 2019-11-06 EP disclosed
US-20190314360-A1 ANTITUMOR AGENT AND BROMODOMAIN INHIBITOR FUJIFILM CORPORATION (JP) 2019-10-17 US disclosed
US-20190314360-A1 ANTITUMOR AGENT AND BROMODOMAIN INHIBITOR FUJIFILM CORPORATION (JP) 2019-10-17 US disclosed
US-20190077761-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND FUJIFILM CORPORATION (JP) 2019-03-14 US disclosed
US-20190077761-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND FUJIFILM CORPORATION (JP) 2019-03-14 US disclosed
EP-3327004-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND Fujifilm Corporation (JP) 2018-05-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10987349-B2 Antitumor agent and bromodomain inhibitor BRD4, BRD1, BRD3 LMNA 1830/4885KDM4E 1027/4885F2 3881/4885
US-10696637-B2 Nitrogen-containing heterocyclic compound CXCL10, CCL5, CXCR3 LMNA 2949/4885KDM4E 3906/4885F2 362/4885
US-20190314360-A1 ANTITUMOR AGENT AND BROMODOMAIN INHIBITOR BRD4, BRD1, BRD3 LMNA 1830/4885KDM4E 1027/4885F2 3881/4885
US-20190077761-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND CXCL10, CCL5, CXCR3 LMNA 2949/4885KDM4E 3906/4885F2 362/4885
US-10633343-B2 CXCL10, CCL5, CXCR3 LMNA 3356/4885KDM4E 3627/4885F2 389/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.