SCHEMBL20184280

SCHEMBL20184280

CC1c2n[nH]c(-c3ccccn3)c2CCN1C=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.37
P2RX7 Q99572 3/20 0.36
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
ALPL P05186 1/20 0.33
PKM P14618 1/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
BTK Q06187 1/20 0.33
PIM1 P11309 3/20 0.32
PRKCQ Q04759 1/20 0.32
PRKCD Q05655 1/20 0.32
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32
DRD3 P35462 1/20 0.32
USP30 Q70CQ3 1/20 0.32
LRRK2 Q5S007 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20184306 0.84 P2RX7 (0.38) P2RX7PIM1
SCHEMBL15019739 0.69 TRPM8 (0.35) PPARG
SCHEMBL16291350 0.65 TACR3 (0.57) P2RX7NPC1SMN1; SMN2
SCHEMBL15020409 0.64 PPARG (0.39) PPARG
SCHEMBL13240633 0.63 KDM4E (0.41) NPC1RAB9ASMN1; SMN2TDP1ALPL
SCHEMBL6968969 0.59 NPC1 (0.48) NPC1RAB9ASMN1; SMN2TDP1ALPL
Dipyridyl SCHEMBL28150180 0.57 KDM4E (0.61) NPC1RAB9ASMN1; SMN2TDP1ALPL
SCHEMBL16200073 0.57 METAP1 (0.44) NPC1RAB9ASMN1; SMN2TDP1ALPL
SCHEMBL21239649 0.56 PARP1 (0.45) P2RX7NPC1SMN1; SMN2
SCHEMBL23199896 0.55 LRRK2 (0.53) NPC1RAB9ASMN1; SMN2TDP1ALPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970267-B3 P2X7 MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-30 EP claimed