SCHEMBL20184677

SCHEMBL20184677

CCc1nc(-c2cccc(C#N)c2)c2c(C(=O)O)c[nH]c2n1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
F11 P03951 1/20 0.43
PIN1 Q13526 1/20 0.43
XDH P47989 1/20 0.43
SLC22A12 Q96S37 1/20 0.43
ADORA2A P29274 3/20 0.43
ADORA2B P29275 2/20 0.43
ADORA1 P30542 2/20 0.43
LRRK2 Q5S007 5/20 0.41
HSP90AB1 P08238 1/20 0.41
IKBKB O14920 3/20 0.40
CHUK O15111 3/20 0.40
ABL1 P00519 1/20 0.40
SGK1 O00141 1/20 0.39
GRIA2 P42262 1/20 0.39
GRIA4 P48058 1/20 0.39
JAK2 O60674 1/20 0.39
JAK3 P52333 1/20 0.39
GRK6 P43250 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20184329 0.87 HSP90AB1 (0.46) HSP90AB1IKBKBCHUKGRIA2GRIA4
SCHEMBL20184548 0.85 JAK3 (0.53) IKBKBCHUKSGK1JAK2JAK3
SCHEMBL20184551 0.85 JAK3 (0.53) PIN1JAK2JAK3
SCHEMBL20184525 0.84 JAK2 (0.49) CHUKSGK1JAK2JAK3
SCHEMBL20184532 0.84 PRKD1 (0.40) HSP90AB1JAK2JAK3
SCHEMBL20184599 0.84 JAK3 (0.53) PIN1HSP90AB1CHUKSGK1JAK2
SCHEMBL20184581 0.84 JAK3 (0.43) JAK2JAK3
SCHEMBL20184478 0.84 JAK2 (0.53) PIN1JAK2JAK3
SCHEMBL20184522 0.84 JAK3 (0.37) LRRK2HSP90AB1IKBKBCHUKJAK2
SCHEMBL20184688 0.83 JAK3 (0.43) JAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2788000-B1 PYRROLOPYRIMIDINES AS JANUS KINASE INHIBITORS MERCK SHARP & DOHME (US) 2018-05-30 EP claimed