SCHEMBL20184548

SCHEMBL20184548

CCc1nc(-c2cccc(O)c2)c2c(C(=O)O)c[nH]c2n1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 11/20 0.53
JAK2 O60674 10/20 0.53
IKBKB O14920 1/20 0.44
CHUK O15111 1/20 0.44
AKR1C3 P42330 1/20 0.42
AKR1C2 P52895 1/20 0.42
AKR1C1 Q04828 1/20 0.42
DHODH Q02127 2/20 0.39
GAA P10253 2/20 0.37
MAPT P10636 2/20 0.37
SGK1 O00141 1/20 0.37
CAMKK2 Q96RR4 1/20 0.37
CHEK1 O14757 1/20 0.37
SIRT5 Q9NXA8 1/20 0.37
TP53 P04637 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20184551 0.89 JAK3 (0.53) JAK3JAK2DHODHMAPTSIRT5
SCHEMBL20184525 0.88 JAK2 (0.49) JAK3JAK2CHUKSGK1CAMKK2
SCHEMBL20184478 0.88 JAK2 (0.53) JAK3JAK2DHODH
SCHEMBL20184599 0.88 JAK3 (0.53) JAK3JAK2CHUKDHODHSGK1
SCHEMBL20184581 0.88 JAK3 (0.43) JAK3JAK2
SCHEMBL20184417 0.87 DYRK1A (0.45) JAK3JAK2DHODHCHEK1
SCHEMBL20184489 0.86 JAK2 (0.51) JAK3JAK2DHODHSGK1CAMKK2
SCHEMBL20184527 0.86 JAK2 (0.49) JAK3JAK2IKBKBCHUKDHODH
SCHEMBL20184518 0.86 PRKAB2 (0.48) JAK3JAK2DHODHMAPT
SCHEMBL20184593 0.86 GPR84 (0.48) JAK3JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2788000-B1 PYRROLOPYRIMIDINES AS JANUS KINASE INHIBITORS MERCK SHARP & DOHME (US) 2018-05-30 EP claimed