SCHEMBL2018490

SCHEMBL2018490

CCn1c(CNC(=O)c2nc(Cl)c(N)nc2N)nc2cc(C(=O)OC)ccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.53
HDAC6 Q9UBN7 1/20 0.46
MAPT P10636 3/20 0.44
NPC1 O15118 2/20 0.44
NLRP3 Q96P20 1/20 0.44
HTT P42858 2/20 0.44
PTGER4 P35408 4/20 0.44
SCNN1A P37088 1/20 0.43
CNR2 P34972 1/20 0.43
NPSR1 Q6W5P4 2/20 0.41
KMT2A Q03164 2/20 0.40
TSHR P16473 2/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
FGB P02675 1/20 0.39
POLB P06746 1/20 0.39
THRB P10828 1/20 0.39
RECQL P46063 1/20 0.39
HSD17B10 Q99714 1/20 0.39
USP2 O75604 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2014471 0.93 MAPT (0.52) KDM4EHDAC6MAPTNPC1NLRP3
SCHEMBL2020165 0.93 ACSS2 (0.46) KDM4EHDAC6HTTSCNN1AKMT2A
SCHEMBL17937045 0.91 HDAC6 (0.43) KDM4EHDAC6MAPTNPC1NLRP3
SCHEMBL2019532 0.91 HDAC6 (0.49) KDM4EHDAC6MAPTHTTSCNN1A
SCHEMBL2019895 0.86 HTT (0.44) HDAC6HTTKMT2ATSHRMEN1
SCHEMBL2021620 0.85 HTT (0.45) KDM4EMAPTNPC1NLRP3HTT
Iodide SCHEMBL2019374 0.85 HTT (0.43) HDAC6HTTKMT2ATSHRMEN1
SCHEMBL2014103 0.85 SCNN1A (0.43) KDM4EHDAC6MAPTNPC1NLRP3
SCHEMBL17937128 0.84 ACSS2 (0.39) KDM4EHDAC6HTTSCNN1A
SCHEMBL2015349 0.83 HTT (0.57) HTTKMT2AMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed