SCHEMBL2020165

SCHEMBL2020165

CCn1c(CNC(=O)c2nc(Cl)c(N)nc2N)nc2ccc(C(=O)OC)cc21

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACSS2 Q9NR19 6/20 0.46
HTT P42858 1/20 0.44
SCNN1A P37088 1/20 0.43
KDM4E B2RXH2 2/20 0.43
TSHR P16473 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP2C9 P11712 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
DRD2 P14416 1/20 0.38
TBXA2R P21731 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2021620 0.93 HTT (0.45) ACSS2HTTKDM4EMEN1KMT2A
SCHEMBL2018490 0.93 KDM4E (0.53) HTTSCNN1AKDM4ETSHRMEN1
SCHEMBL2017836 0.91 HTT (0.46) ACSS2HTTSCNN1AMEN1KMT2A
SCHEMBL12635756 0.90 HTT (0.49) ACSS2HTTTSHRMEN1KMT2A
SCHEMBL2019384 0.90 HTT (0.41) ACSS2HTTSCNN1AKDM4ETSHR
SCHEMBL2015541 0.89 HTT (0.46) ACSS2HTTTSHR
SCHEMBL2020396 0.88 HTT (0.48) ACSS2HTTMEN1KMT2AHDAC6
SCHEMBL2018438 0.88 SCNN1A (0.44) ACSS2HTTSCNN1A
SCHEMBL2040435 0.88 HTT (0.45) ACSS2HTTTSHRMEN1KMT2A
SCHEMBL2016331 0.87 HTT (0.52) ACSS2HTTSCNN1AKDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed