SCHEMBL2014471

SCHEMBL2014471

CCOC(=O)c1ccc2c(c1)nc(CNC(=O)c1nc(Cl)c(N)nc1N)n2CC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.52
NPC1 O15118 2/20 0.52
NLRP3 Q96P20 1/20 0.52
NPSR1 Q6W5P4 2/20 0.50
HTT P42858 2/20 0.47
HSD17B10 Q99714 1/20 0.47
ALDH1A1 P00352 5/20 0.47
HPGD P15428 3/20 0.47
KMT2A Q03164 3/20 0.46
RAB9A P51151 2/20 0.46
MEN1 O00255 2/20 0.46
KDM4E B2RXH2 1/20 0.46
ATM Q13315 1/20 0.45
HDAC6 Q9UBN7 1/20 0.44
GAA P10253 1/20 0.43
SIRT2 Q8IXJ6 1/20 0.42
SIRT1 Q96EB6 1/20 0.42
RECQL P46063 1/20 0.42
PTGER4 P35408 2/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2021620 0.93 HTT (0.45) MAPTNPC1NLRP3NPSR1HTT
SCHEMBL2018490 0.93 KDM4E (0.53) MAPTNPC1NLRP3NPSR1HTT
SCHEMBL17937045 0.90 HDAC6 (0.43) MAPTNPC1NLRP3NPSR1HTT
SCHEMBL2019532 0.89 HDAC6 (0.49) MAPTHTTHSD17B10ALDH1A1HPGD
SCHEMBL2020165 0.85 ACSS2 (0.46) HTTALDH1A1KMT2AMEN1KDM4E
SCHEMBL2019384 0.84 HTT (0.41) MAPTNPC1NLRP3NPSR1HTT
SCHEMBL2019895 0.84 HTT (0.44) HTTHSD17B10KMT2AMEN1HDAC6
Iodide SCHEMBL2019374 0.83 HTT (0.43) HTTHSD17B10KMT2AMEN1HDAC6
SCHEMBL2015349 0.82 HTT (0.57) HTTHPGDKMT2AMEN1GAA
SCHEMBL2016173 0.82 HTT (0.42) HTTHSD17B10ALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed