SCHEMBL20188096

SCHEMBL20188096

C=CCOc1cc(C(C)N)ccc1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 12/20 0.42
HTR2B P41595 8/20 0.42
HTR2A P28223 7/20 0.39
ADRB2 P07550 3/20 0.39
HTR1A P08908 3/20 0.39
SLC6A4 P31645 3/20 0.39
CHRM5 P08912 2/20 0.39
ADRA2A P08913 2/20 0.39
DRD2 P14416 2/20 0.39
ADRA2B P18089 2/20 0.39
ADRA2C P18825 2/20 0.39
DRD4 P21917 2/20 0.39
HRH2 P25021 2/20 0.39
HTR7 P34969 2/20 0.39
DRD3 P35462 2/20 0.39
HTR6 P50406 2/20 0.39
KCNH2 Q12809 2/20 0.39
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
SLC22A1 O15245 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18374457 1.00 HTR2C (0.42) HTR2CHTR2BHTR2AADRB2HTR1A
Hydrochloric Acid SCHEMBL20338513 0.98 HTR2C (0.43) HTR2CHTR2BHTR2AADRB2HTR1A
Hydrochloric Acid SCHEMBL20338511 0.98 HTR2C (0.43) HTR2CHTR2BHTR2AADRB2HTR1A
SCHEMBL20206848 0.88 ACHE (0.41) HTR2CHTR2BHTR2AADRB2HTR1A
SCHEMBL20206845 0.82 HTR2C (0.38) HTR2CHTR2BHTR2AADRB2HTR1A
SCHEMBL31447482 0.81 HTT (0.44) ADRB2TSHRLMNAMAPTALDH1A1
SCHEMBL28408399 0.81 HTT (0.44) ADRB2TSHRLMNAMAPTALDH1A1
SCHEMBL20201941 0.80 ALDH1A1 (0.44) ADRB2GAAALDH1A1
SCHEMBL18374263 0.78 MAPT (0.39) HTR2CHTR2BHTR2AADRB2GAA
SCHEMBL12094250 0.78 DUT (0.41) HTR2CHTR2BHTR2AADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018128720-A1 URACIL CONTAINING COMPOUNDS CV6 THERAPEUTICS (NI) LIMITED (GB) 2018-07-12 WO disclosed
WO-2018098207-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2018-05-31 WO disclosed