SCHEMBL2019384

SCHEMBL2019384

CCCCOC(=O)c1ccc2nc(CNC(=O)c3nc(Cl)c(N)nc3N)n(CC)c2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.41
TP53 P04637 2/20 0.39
S1PR3 Q99500 1/20 0.39
ACSS2 Q9NR19 3/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
PDE4D Q08499 1/20 0.38
MAPT P10636 2/20 0.37
NPC1 O15118 1/20 0.37
NLRP3 Q96P20 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
SCNN1A P37088 4/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2021620 0.91 HTT (0.45) HTTS1PR3ACSS2MAPTNPC1
SCHEMBL2020165 0.90 ACSS2 (0.46) HTTACSS2CYP2C9TSHRMEN1
SCHEMBL2017836 0.86 HTT (0.46) HTTTP53ACSS2LMNAMEN1
SCHEMBL12635756 0.85 HTT (0.49) HTTACSS2TSHRMEN1KMT2A
SCHEMBL2014471 0.84 MAPT (0.52) HTTTSHRMAPTNPC1NLRP3
SCHEMBL2018430 0.84 ACSS2 (0.42) HTTS1PR3ACSS2MEN1KMT2A
SCHEMBL2020396 0.84 HTT (0.48) HTTTP53ACSS2LMNAMEN1
SCHEMBL2018438 0.83 SCNN1A (0.44) HTTTP53ACSS2MAPTSCNN1A
SCHEMBL2015541 0.83 HTT (0.46) HTTACSS2TSHR
SCHEMBL2040435 0.83 HTT (0.45) HTTTP53ACSS2LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed