SCHEMBL2020148

SCHEMBL2020148

CC(C(N)=O)N(C)Cc1ccc(OCc2cccc(Cl)c2)cc1

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAOB P27338 8/20 0.62
ALOX5 P09917 1/20 0.61
MAOA P21397 3/20 0.56
RXRA P19793 1/20 0.54
RXRB P28702 1/20 0.54
RXRG P48443 1/20 0.54
ADAMTS4 O75173 1/20 0.49
MMP13 P45452 1/20 0.49
FFAR1 O14842 1/20 0.49
PKM P14618 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2020147 1.00 MAOB (0.62) MAOBALOX5MAOARXRARXRB
SCHEMBL7396817 0.87 MAOB (0.60) MAOBALOX5MAOARXRARXRB
SCHEMBL9131943 0.87 MAOB (0.60) MAOBALOX5MAOARXRARXRB
SCHEMBL9129876 0.86 MAOB (0.71) MAOBMAOA
SCHEMBL7396562 0.86 MAOB (0.71) MAOBMAOA
SCHEMBL1071203 0.86 MAOB (0.58) MAOBALOX5MAOAFFAR1
SCHEMBL8935317 0.83 ALOX5 (0.62) MAOBALOX5MAOARXRARXRB
SCHEMBL9516428 0.82 MAOB (0.53) MAOBALOX5MAOAFFAR1
SCHEMBL9126134 0.82 MAOB (0.53) MAOBALOX5MAOAFFAR1
SCHEMBL2017533 0.81 ALOX5 (0.63) MAOBALOX5MAOARXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110160308-A1 Use of Monoamine Oxidase Inhibitors to Treat Outer Retina Disorders ALCON RESEARCH, LTD. (US) 2011-06-30 US disclosed
CN-101495185-A Monoamine oxidase inhibitors for the treatment of disorders of the outer retina ALCON RES LTD (US) 2009-07-29 CN disclosed
EP-0400495-B1 N-phenylalkyl substituted alpha-amino carboxamide derivatives and process for their preparation. ERBA CARLO SPA (IT) 1993-11-03 EP disclosed
EP-0426816-A1 N-PHENYLALKYL SUBSTITUTED $g(a)-AMINO CARBOXAMIDE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-05-15 EP disclosed
EP-0400495-A1 N-phenylalkyl substituted alfa-amino carboxamide derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1990-12-05 EP disclosed
WO-1990014334-A1 N-PHENYLALKYL SUBSTITUTED α-AMINO CARBOXAMIDE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.R.L. (IT) 1990-11-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110160308-A1 Use of Monoamine Oxidase Inhibitors to Treat Outer Retina Disorders MAOB, MAOA, ALDH1A2 MAOB 1/4885ALOX5 397/4885MAOA 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.