SCHEMBL20203378

SCHEMBL20203378

C=CC1(C)CC(c2ccc(Cl)cc2)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP1LC3B Q9GZQ8 1/20 0.38
HTR3A P46098 1/20 0.38
KDM1A O60341 2/20 0.38
RCOR1 Q9UKL0 2/20 0.38
DRD2 P14416 1/20 0.38
SRD5A1 P18405 2/20 0.36
SLC6A3 Q01959 2/20 0.35
SLC6A2 P23975 1/20 0.35
MAPK1 P28482 1/20 0.35
LIG1 P18858 1/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
ALOX12 P18054 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
LSS P48449 1/20 0.33
SLC2A1 P11166 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL11481432 0.70 MAPK1 (0.49) MAP1LC3BHTR3AKDM1ARCOR1DRD2
SCHEMBL11481127 0.69 MAPK1 (0.47) MAP1LC3BHTR3ASRD5A1SLC6A3MAPK1
SCHEMBL4339855 0.67 KDM1A (0.53) KDM1ARCOR1MAPK1LIG1MEN1
SCHEMBL30074982 0.66 TRPA1 (0.47) HTR3AKDM1ARCOR1DRD2SRD5A1
SCHEMBL1858459 0.66 HTR3A (0.37) MAP1LC3BHTR3AKDM1ARCOR1DRD2
SCHEMBL31622423 0.65 HTR3A (0.48) HTR3AKDM1ARCOR1DRD2SLC6A3
SCHEMBL27276966 0.65 KDM1A (0.43) HTR3AKDM1ARCOR1DRD2SRD5A1
SCHEMBL19502447 0.65 HTR3A (0.44) MAP1LC3BHTR3ADRD2SRD5A1SLC6A3
SCHEMBL315186 0.65 HTR3A (0.58) HTR3ADRD2SRD5A1SLC6A3SLC6A2
Methyl Alcohol SCHEMBL15391253 0.65 DRD2 (0.55) HTR3ADRD2SRD5A1SLC6A3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3544979-B1 OXADIAZOLONES AS TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS HOFFMANN LA ROCHE (CH) 2021-08-04 EP disclosed
WO-2018096159-A1 OXADIAZOLONES AS TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2018-05-31 WO disclosed