SCHEMBL20215264

SCHEMBL20215264

CS(=O)(=O)c1ccc(Cn2ccc(=O)cc2-c2cccc(C(F)(F)F)c2Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.43
FLT3 P36888 1/20 0.36
PTGS2 P35354 3/20 0.35
CHRM5 P08912 1/20 0.35
CHRM3 P20309 1/20 0.35
MAPT P10636 1/20 0.35
ALDH1A1 P00352 3/20 0.35
ALDH2 P05091 3/20 0.35
ALDH3A1 P30838 3/20 0.35
SDHB P21912 2/20 0.35
KIF11 P52732 1/20 0.34
RORC P51449 1/20 0.34
NR1H2 P55055 3/20 0.34
NR1H3 Q13133 3/20 0.34
NR3C2 P08235 1/20 0.34
NOTUM Q6P988 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20215232 0.87 MAPT (0.47) P2RX7MAPTNOTUM
SCHEMBL20215244 0.87 MAPT (0.39) P2RX7CHRM5CHRM3MAPTALDH1A1
SCHEMBL20215217 0.86 P2RX7 (0.43) P2RX7CHRM5CHRM3MAPTALDH1A1
SCHEMBL20215257 0.86 CHRM5 (0.46) P2RX7CHRM5CHRM3MAPTALDH1A1
SCHEMBL20215219 0.86 P2RX7 (0.41) P2RX7MAPTALDH1A1NOTUM
SCHEMBL20215242 0.84 MAPT (0.46) P2RX7CHRM5MAPT
SCHEMBL20215246 0.84 PPARG (0.37) P2RX7CHRM5ALDH1A1NOTUM
SCHEMBL20215231 0.83 MAPT (0.46) P2RX7MAPTALDH1A1
SCHEMBL20215256 0.83 KDM4E (0.43) P2RX7MAPTALDH1A1
SCHEMBL20215254 0.82 HCRTR1 (0.41) P2RX7CHRM5CHRM3MAPTNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9988373-B2 Nitrogen-containing six-membered cyclic derivatives and pharmaceutical composition comprising the same SHIONOGI & CO., LTD. (JP) 2018-06-05 US disclosed
US-9988373-B2 Nitrogen-containing six-membered cyclic derivatives and pharmaceutical composition comprising the same SHIONOGI & CO., LTD. (JP) 2018-06-05 US disclosed