SCHEMBL20217431

SCHEMBL20217431

CN1CCC(Oc2ccc(C(=N)c3cc(NC(=O)C(c4ccccn4)C4CCCC4)ccc3N)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.41
DYRK1A Q13627 9/20 0.40
CLK2 P49760 2/20 0.40
CLK3 P49761 2/20 0.40
ROCK2 O75116 1/20 0.39
CYP3A4 P08684 1/20 0.39
TTK P33981 1/20 0.39
AURKB Q96GD4 1/20 0.39
INCENP Q9NQS7 1/20 0.39
GSK3B P49841 8/20 0.39
F10 P00742 2/20 0.38
F2 P00734 1/20 0.38
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
F7 P08709 1/20 0.38
F3 P13726 1/20 0.38
PRSS3 P35030 1/20 0.38
GRM4 Q14833 1/20 0.37
LCK P06239 1/20 0.36
MAPK14 Q16539 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20217530 0.86 KDR (0.40) KDRDYRK1ACLK2CLK3GSK3B
SCHEMBL20217416 0.86 KDR (0.41) KDRDYRK1ACLK2CLK3F10
SCHEMBL20217632 0.84 CYP3A4 (0.52) KDRCYP3A4TTKAURKBINCENP
SCHEMBL20217315 0.83 CYP3A4 (0.52) KDRCYP3A4TTKAURKBINCENP
SCHEMBL20217450 0.81 CYP3A4 (0.42) KDRROCK2CYP3A4TTKAURKB
SCHEMBL20217751 0.81 CYP3A4 (0.55) KDRCYP3A4TTKAURKBINCENP
SCHEMBL20217430 0.81 F10 (0.42) KDRDYRK1ACLK2CLK3F10
SCHEMBL20217418 0.80 FFAR2 (0.45) KDRGRM4LMNAMEN1HTR1E
SCHEMBL15477042 0.79 CYP3A4 (0.55) DYRK1ACLK2CLK3ROCK2CYP3A4
SCHEMBL20217405 0.77 MAPT (0.44) KDRROCK2F10LCKLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2766352-B1 INDAZOLE COMPOUNDS AS KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIV HEALTH NETWORK UHN (CA) 2018-06-06 EP disclosed