SCHEMBL20217586

SCHEMBL20217586

CCCC(C)CC(CC(C)C)Nc1ccc(C(=N)c2cc(C(=O)NC(c3ccccn3)C(C)C)ccc2N)cc1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 7/20 0.35
TAS1R1 Q7RTX1 7/20 0.35
F7 P08709 3/20 0.34
TEAD4 Q15561 1/20 0.33
F3 P13726 4/20 0.32
S1PR2 O95136 1/20 0.31
S1PR4 O95977 1/20 0.31
S1PR3 Q99500 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LNPEP Q9UIQ6 1/20 0.31
ERAP2 Q6P179 1/20 0.31
F2 P00734 1/20 0.30
F10 P00742 1/20 0.30
PRSS1 P07477 1/20 0.30
PRSS2 P07478 1/20 0.30
PRSS3 P35030 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20217678 0.75 ALDH1A1 (0.38) F7S1PR2S1PR4S1PR3ALDH1A1
SCHEMBL20217652 0.75 TAS1R3 (0.40) TAS1R3TAS1R1F7F3S1PR2
SCHEMBL20217171 0.70 CYP3A4 (0.43) TAS1R3TAS1R1F7F3S1PR2
SCHEMBL20217231 0.70 CYP3A4 (0.43) TAS1R3TAS1R1F7F3S1PR2
SCHEMBL20217664 0.70 CYP3A4 (0.47) ALDH1A1
SCHEMBL20217358 0.70 ACACB (0.38) ALDH1A1LNPEP
SCHEMBL20217478 0.68 LMNA (0.42) ALDH1A1
SCHEMBL20217669 0.67 MEN1 (0.40) TAS1R3TAS1R1ALDH1A1F10
SCHEMBL20217428 0.67 CYP3A4 (0.41) F7
SCHEMBL20217912 0.66 CYP3A4 (0.43) S1PR2S1PR4S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2766352-B1 INDAZOLE COMPOUNDS AS KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIV HEALTH NETWORK UHN (CA) 2018-06-06 EP disclosed