SCHEMBL20217652

SCHEMBL20217652

CCCc1ccc(C(=N)c2cc(C(=O)NC(CC(C)C)c3ccccn3)ccc2N)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.40
TAS1R1 Q7RTX1 2/20 0.40
CYP3A4 P08684 1/20 0.40
TTK P33981 1/20 0.40
AURKB Q96GD4 1/20 0.40
INCENP Q9NQS7 1/20 0.40
TACR3 P29371 1/20 0.37
F2 P00734 1/20 0.37
F10 P00742 1/20 0.37
F7 P08709 1/20 0.37
F3 P13726 1/20 0.37
PPARG P37231 1/20 0.36
NR2F2 P24468 1/20 0.36
PAX8 Q06710 1/20 0.36
KLF5 Q13887 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
BDKRB2 P30411 1/20 0.35
S1PR2 O95136 1/20 0.35
S1PR4 O95977 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20217231 0.85 CYP3A4 (0.43) TAS1R3TAS1R1CYP3A4TTKAURKB
SCHEMBL20217171 0.85 CYP3A4 (0.43) TAS1R3TAS1R1CYP3A4TTKAURKB
SCHEMBL20217438 0.78 KDM4E (0.50) CYP3A4L3MBTL1NPC1POLBRAB9A
SCHEMBL20217226 0.77 CYP3A4 (0.44) TAS1R3TAS1R1CYP3A4TTKAURKB
SCHEMBL20217586 0.75 TAS1R3 (0.35) TAS1R3TAS1R1F2F10F7
SCHEMBL20217912 0.71 CYP3A4 (0.43) CYP3A4TTKAURKBINCENPS1PR2
SCHEMBL20217678 0.70 ALDH1A1 (0.38) CYP3A4TTKAURKBINCENPF2
SCHEMBL20217347 0.70 ALDH1A1 (0.47) TAS1R3TAS1R1PPARGLMNA
SCHEMBL20217403 0.70 TAS1R3 (0.43) TAS1R3TAS1R1PPARGLMNA
SCHEMBL20217428 0.69 CYP3A4 (0.41) CYP3A4TTKAURKBINCENPF7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2766352-B1 INDAZOLE COMPOUNDS AS KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIV HEALTH NETWORK UHN (CA) 2018-06-06 EP disclosed