SCHEMBL20217587

SCHEMBL20217587

CC(C)CC(C)NC(=O)c1ccc(N)c(C(=N)c2ccc(N3C4CCC3CC(O)C4)cc2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.37
TTK P33981 1/20 0.37
AURKB Q96GD4 1/20 0.37
INCENP Q9NQS7 1/20 0.37
MLYCD O95822 1/20 0.36
ITGB3 P05106 6/20 0.34
ITGA2B P08514 6/20 0.34
SMYD3 Q9H7B4 2/20 0.32
HSP90AA1 P07900 3/20 0.31
HSP90AB1 P08238 3/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
CHRM2 P08172 1/20 0.31
CTSK P43235 1/20 0.31
ERAP2 Q6P179 1/20 0.31
ERAP1 Q9NZ08 1/20 0.31
LNPEP Q9UIQ6 1/20 0.31
F2 P00734 1/20 0.31
F10 P00742 1/20 0.31
PRSS1 P07477 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20217341 0.78 CYP3A4 (0.40) CYP3A4TTKAURKBINCENPSMYD3
SCHEMBL20217636 0.76 NAMPT (0.39) HSP90AA1HSP90AB1
SCHEMBL20217804 0.76 RAB9A (0.43) CYP3A4TTKAURKBINCENPNPC1
SCHEMBL20217529 0.72 L3MBTL1 (0.45) CYP3A4RAB9A
SCHEMBL20217764 0.69 CYP3A4 (0.49) CYP3A4TTKAURKBINCENPF2
SCHEMBL20217496 0.67 CYP3A4 (0.62) CYP3A4TTKAURKBINCENPF2
SCHEMBL20217662 0.67 CYP3A4 (0.47) CYP3A4TTKAURKBINCENPSMYD3
SCHEMBL20217579 0.67 CYP3A4 (0.65) CYP3A4TTKAURKBINCENP
SCHEMBL20217956 0.67 CYP3A4 (0.48) CYP3A4TTKAURKBINCENPSMYD3
SCHEMBL20217623 0.67 HPGD (0.45) NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2766352-B1 INDAZOLE COMPOUNDS AS KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIV HEALTH NETWORK UHN (CA) 2018-06-06 EP disclosed