SCHEMBL202480

SCHEMBL202480

O=[N+]([O-])c1c(Cl)cnc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
S100A4 P26447 1/20 0.44
ALDH1A1 P00352 6/20 0.44
POLB P06746 1/20 0.44
MAPT P10636 4/20 0.43
CYP3A4 P08684 1/20 0.42
KDM4E B2RXH2 4/20 0.41
TDP1 Q9NUW8 1/20 0.41
GPR3 P46089 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
NPSR1 Q6W5P4 2/20 0.39
LMNA P02545 1/20 0.39
XBP1 P17861 1/20 0.39
PAX8 Q06710 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561101 0.81 POLB (0.53) MEN1KMT2AS100A4ALDH1A1POLB
SCHEMBL8568380 0.79 MEN1 (0.45) MEN1KMT2AS100A4ALDH1A1POLB
SCHEMBL31581131 0.79 MEN1 (0.45) MEN1KMT2AS100A4ALDH1A1POLB
SCHEMBL9602589 0.79 S100A4 (0.53) MEN1KMT2AS100A4ALDH1A1POLB
SCHEMBL2004290 0.78 POLB (0.54) MEN1KMT2AALDH1A1POLBMAPT
SCHEMBL203184 0.78 PTGES (0.44) ALDH1A1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL8566835 0.77 MEN1 (0.43) MEN1KMT2AS100A4ALDH1A1POLB
SCHEMBL202663 0.76 POLB (0.51) MEN1KMT2AALDH1A1POLBMAPT
SCHEMBL29381779 0.76 POLB (0.51) MEN1KMT2AALDH1A1POLBMAPT
SCHEMBL21632211 0.76 CYP3A4 (0.50) MEN1KMT2AALDH1A1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112624970-B Application of 8-bit aryl substituted quinoline nitrogen oxide in plant virus resistance and sterilization 南开大学 2022-10-28 CN disclosed
CN-112624970-A Application of 8-bit aryl substituted quinoline nitrogen oxide in plant virus resistance and sterilization 南开大学 2021-04-09 CN disclosed
US-8546383-B2 Chiral fused [1,2]imidazo[4,5-c] ring compounds 3M INNOVATIVE PROPERTIES COMPANY (US) 2013-10-01 US disclosed
CN-103232461-A Synthesis method of 4-chloroquine anhydride SUZHOU KEJIE BIOLOG PHARMACEUTICAL CO LTD 2013-08-07 CN disclosed
US-20120232057-A1 CHIRAL FUSED [1,2]IMIDAZO[4,5-c] RING COMPOUNDS 3M INNOVATIVE PROPERTIES COMPANY 2012-09-13 US disclosed
EP-1831226-B1 CHIRAL TETRACYCLIC COMPOUNDS INDUCING INTERFERON BIOSYNTHESIS 3M INNOVATIVE PROPERTIES CO (US) 2012-08-08 EP disclosed
US-8207162-B2 Chiral fused [1,2]imidazo[4,5-c] ring compounds 3M INNOVATIVE PROPERTIES COMPANY (US) 2012-06-26 US disclosed
US-8088788-B2 Substituted fused[1,2] imidazo[4,5-c] ring compounds and methods 3M INNOVATIVE PROPERTIES COMPANY (US) 2012-01-03 US disclosed
US-20110207725-A1 CHIRAL FUSED [1,2]IMIDAZO[4,5-c] RING COMPOUNDS 3M INNOVATIVE PROPERTIES COMPANY 2011-08-25 US disclosed
US-7943609-B2 Such as (tetrahydr)imidazo(4,5-c ) quinoline or naphthymidine; immunomoderators; induce cytokine biosynthesis in animals; anticancer agents; viricides 3M INNOVATIVE PROPRERTIES COMPANY (US) 2011-05-17 US disclosed
CN-101823996-A Preparation method of 2,8-bit acyl substituted quinoline ASTA CHENGDU BIO PHARMACEUTICAL CO LTD 2010-09-08 CN disclosed
CN-101823997-A Preparation method of 2-bit acyl substituted quinoline ASTA CHENGDU BIO PHARMACEUTICAL CO LTD 2010-09-08 CN disclosed
US-20090221551-A1 SUBSTITUTED FUSED[1,2] IMIDAZO[4,5C] RING COMPOUNDS AND METHODS PFIZER INC. 2009-09-03 US disclosed
EP-1831226-A4 CHIRAL FUSED 1,2 IMIDAZO 4,5-c RING COMPOUNDS 3M INNOVATIVE PROPERTIES CO (US) 2008-11-05 EP disclosed
US-20080269192-A1 Chiral Fused [1,2]Imidazo[4,5-C] Ring Compounds COLEY PHARMACEUTICAL GROUP, INC. (US) 2008-10-30 US disclosed
US-20080070907-A1 Substituted chiral fused [1,2] imidazo [4,5-C] ring compounds and methods COLEY PHARMACEUTICAL GROUP, INC. (US) 2008-03-20 US disclosed
WO-2008008432-A2 SUBSTITUTED CHIRAL FUSED( 1,2) IMIDAZO (4,5-C) RING COMPOUNDS AND METHODS COLEY PHARMACEUTICAL GROUP, INC. (US) 2008-01-17 WO disclosed
WO-2007106852-A2 SUBSTITUTED FUSED[1,2]IMIDAZO[4,5-C] RING COMPOUNDS AND METHODS COLEY PHARMACEUTICAL GROUP, INC. (US) 2007-09-20 WO disclosed
EP-1831226-A2 CHIRAL FUSED 1,2 IMIDAZO 4,5-c RING COMPOUNDS 3M INNOVATIVE PROPERTIES COMPANY (US) 2007-09-12 EP disclosed
WO-2006074003-A2 CHIRAL FUSED [1,2]IMIDAZO[4,5-c] RING COMPOUNDS 3M INNOVATIVE PROPERTIES COMPANY (US) 2006-07-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080269192-A1 Chiral Fused [1,2]Imidazo[4,5-C] Ring Compounds IFNAR1, IFNG, IL4 MEN1 2108/4885KMT2A 3480/4885S100A4 1803/4885
US-20120232057-A1 CHIRAL FUSED [1,2]IMIDAZO[4,5-c] RING COMPOUNDS IFNAR1, IFNG, IL4 MEN1 2062/4885KMT2A 3459/4885S100A4 1794/4885
US-20110207725-A1 CHIRAL FUSED [1,2]IMIDAZO[4,5-c] RING COMPOUNDS IFNAR1, IFNG, IL4 MEN1 2108/4885KMT2A 3480/4885S100A4 1803/4885
US-20080070907-A1 Substituted chiral fused [1,2] imidazo [4,5-C] ring compounds and methods IFNAR1, IL2, IFNG MEN1 2993/4885KMT2A 3186/4885S100A4 1787/4885
US-20090221551-A1 SUBSTITUTED FUSED[1,2] IMIDAZO[4,5C] RING COMPOUNDS AND METHODS IL2, IFNG, IL4 MEN1 4112/4885KMT2A 3293/4885S100A4 1530/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.