SCHEMBL20255376

SCHEMBL20255376

Cc1ccc2c(c1)CNCC(C)(C)C2

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.35
HTR5A P47898 3/20 0.33
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
METAP1 P53582 1/20 0.32
PARP10 Q53GL7 2/20 0.31
PARP11 Q9NR21 1/20 0.31
PARP1 P09874 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18734225 0.81
SCHEMBL11530207 0.78 ADRA2A (0.41) ADRA2AHTR5AMETAP1ALDH1A1CYP3A4
SCHEMBL18322409 0.77 PNMT (0.43) HTR2AHTR2CHTR2BALDH1A1
SCHEMBL11988468 0.76 HTR2A (0.40) ADRA2AHTR5AHTR2AHTR2CHTR2B
SCHEMBL30560114 0.76 CHRNB2 (0.41) ADRA2AHTR5AMETAP1PARP10PARP11
SCHEMBL5068876 0.76 CHRNB2 (0.41) ADRA2AHTR5AMETAP1PARP10PARP11
Hydrochloric Acid SCHEMBL18706568 0.76 PNMT (0.42) HTR2AHTR2CHTR2BALDH1A1
Hydrochloric Acid SCHEMBL3118573 0.74 CHRNB2 (0.39) ADRA2AHTR5AMETAP1PARP10PARP11
SCHEMBL14886110 0.71 ADRA2A (0.38) ADRA2AHTR5AHTR2AHTR2CHTR2B
SCHEMBL22549228 0.71 HTR5A (0.33) ADRA2AHTR5AMETAP1PARP10PARP11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018104766-A1 3-(2,3-DIHYDRO-1H-INDEN-5-YL)PROPANOIC ACID DERIVATIVES AND THEIR USE AS NRF2 REGULATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-06-14 WO disclosed