SCHEMBL2025839

SCHEMBL2025839

CCCCOC(=O)N1CCC(c2ccc(N)cc2)C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 4/20 0.53
PRMT5 O14744 5/20 0.51
WDR77 Q9BQA1 5/20 0.51
LMNA P02545 4/20 0.50
CYP1A2 P05177 2/20 0.50
CYP3A4 P08684 2/20 0.50
CYP2C9 P11712 1/20 0.50
TSHR P16473 1/20 0.50
CYP2C19 P33261 1/20 0.50
PDE4D Q08499 1/20 0.50
MAPT P10636 2/20 0.45
RAB9A P51151 2/20 0.45
ALDH1A1 P00352 2/20 0.45
NPC1 O15118 1/20 0.45
POLB P06746 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CHRM2 P08172 1/20 0.41
HTR1A P08908 1/20 0.41
GAA P10253 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23040449 0.94 LMNA (0.49) PDE4BPRMT5WDR77LMNACYP1A2
SCHEMBL30376364 0.93 LMNA (0.49) PDE4BPRMT5WDR77LMNACYP1A2
SCHEMBL31455322 0.90 LMNA (0.51) PDE4BPRMT5WDR77LMNACYP1A2
SCHEMBL4709679 0.88 PRMT5 (0.64) PDE4BPRMT5WDR77LMNACYP1A2
SCHEMBL22659030 0.85 PDE4B (0.53) PDE4BPRMT5WDR77LMNAPDE4D
SCHEMBL15531501 0.83 LMNA (0.50) PDE4BLMNACYP1A2CYP3A4CYP2C9
SCHEMBL2047643 0.83 LMNA (0.45) PDE4BPRMT5WDR77LMNACYP1A2
SCHEMBL2023788 0.82 LMNA (0.49) PDE4BPRMT5WDR77LMNACYP1A2
SCHEMBL29742014 0.80 TRPC6 (0.50) PDE4BLMNARAB9AALDH1A1NPC1
SCHEMBL15379831 0.80 LMNA (0.49) LMNACYP1A2CYP3A4CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2516392-A1 SUBSTITUTED BENZAMIDE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2012-10-31 EP disclosed
WO-2011076678-A1 SUBSTITUTED BENZAMIDE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-06-30 WO disclosed