SCHEMBL20260918

SCHEMBL20260918

Cc1c(Nc2ncn(-c3cc(F)cc(F)c3)n2)cccc1N1CCN(C2COC2)CC1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CSNK2A2 P19784 2/20 0.36
CSNK2A1 P68400 2/20 0.36
BTK Q06187 2/20 0.35
ATR Q13535 3/20 0.35
LRRK2 Q5S007 2/20 0.35
KCNH2 Q12809 1/20 0.35
JAK2 O60674 2/20 0.34
PTK2 Q05397 2/20 0.33
TBK1 Q9UHD2 2/20 0.33
SYK P43405 1/20 0.33
PRKDC P78527 1/20 0.32
MGLL Q99685 2/20 0.32
HTR1A P08908 1/20 0.32
MAPK8 P45983 1/20 0.32
MAPK10 P53779 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18278231 0.88 LRRK2 (0.35) CSNK2A2CSNK2A1BTKATRLRRK2
SCHEMBL20260920 0.87 GAA (0.41) MAPK8MAPK10
SCHEMBL20260924 0.86 MAPK8 (0.35) MAPK8MAPK10
SCHEMBL18278381 0.84 LRRK2 (0.35) CSNK2A2CSNK2A1ATRLRRK2KCNH2
SCHEMBL20260546 0.84 P2RX7 (0.37) ATRJAK2PTK2TBK1SYK
SCHEMBL18277832 0.83 ATR (0.35) CSNK2A2CSNK2A1BTKATRLRRK2
SCHEMBL20260877 0.83 TBK1 (0.43) JAK2PTK2TBK1MAPK8MAPK10
SCHEMBL20260500 0.83 TBK1 (0.34) CSNK2A2CSNK2A1ATRLRRK2KCNH2
SCHEMBL20260507 0.83 TBK1 (0.38) JAK2PTK2TBK1MAPK8MAPK10
SCHEMBL18278671 0.81 ATR (0.35) CSNK2A2CSNK2A1ATRLRRK2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018106646-A1 AMINOTRIAZOLES FOR THE TREATMENT OF DEMYELINATING DISEASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2018-06-14 WO disclosed