SCHEMBL20274221

SCHEMBL20274221

O=C(CO)N1CCN(C(=O)c2nc3cc(C(F)(F)F)ccc3s2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.46
RBP4 P02753 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HPGD P15428 1/20 0.44
RAB9A P51151 1/20 0.44
ALOX5 P09917 1/20 0.44
AKR1B1 P15121 6/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HRH4 Q9H3N8 1/20 0.41
TRPV1 Q8NER1 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
AKR1A1 P14550 1/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL604903 0.86 HRH4 (0.56) DYRK1ARBP4SMN1; SMN2HPGDRAB9A
SCHEMBL20274141 0.84 RAB9A (0.52) DYRK1ARAB9A
SCHEMBL28222855 0.84 SCN9A (0.48) DYRK1ARBP4SMN1; SMN2HPGDRAB9A
SCHEMBL20274125 0.82 AKR1B1 (0.53) DYRK1AAKR1B1TRPV1AKR1A1
SCHEMBL20274202 0.80 AKR1B1 (0.50) DYRK1ASMN1; SMN2HPGDALOX5AKR1B1
Lithium Ion SCHEMBL31084584 0.75 DYRK1A (0.56) DYRK1AALOX5AKR1B1TRPV1MEN1
SCHEMBL3613102 0.75 DYRK1A (0.56) DYRK1AALOX5AKR1B1TRPV1MEN1
SCHEMBL3642935 0.75 DYRK1A (0.58) DYRK1AALOX5AKR1B1TRPV1MEN1
SCHEMBL3613098 0.73 DYRK1A (0.57) DYRK1AALOX5AKR1B1TRPV1MEN1
SCHEMBL20274138 0.71 FAAH (0.46) ALOX5PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2922845-B1 ANTHELMINTIC COMPOUNDS AND COMPOSITIONS AND METHOD OF USING THEREOF MERIAL INC (US) 2018-06-20 EP disclosed