SCHEMBL20311540

SCHEMBL20311540

NNc1ccc(NN)c(N)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
IDO1 P14902 1/20 0.36
CYP2C19 P33261 1/20 0.36
PTGS2 P35354 1/20 0.36
KDM4E B2RXH2 9/20 0.35
MAPT P10636 8/20 0.35
NPC1 O15118 2/20 0.35
POLB P06746 1/20 0.35
RAB9A P51151 1/20 0.35
GAA P10253 7/20 0.33
GFER P55789 5/20 0.33
CA1 P00915 3/20 0.33
CA2 P00918 3/20 0.33
CA9 Q16790 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21646381 0.84 PRKCI (0.40) TDP1KDM4EMAPTNPC1GAA
SCHEMBL4167680 0.79 TDP1 (0.39) TDP1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL12287691 0.79 TDP1 (0.46) TDP1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL7589418 0.77 CASP1 (0.44) TDP1CYP3A4KDM4EMAPTNPC1
Hydrochloric Acid SCHEMBL28937662 0.75 CASP1 (0.42) TDP1CYP3A4KDM4EMAPTNPC1
SCHEMBL14218921 0.73 TDP1 (0.54) TDP1CYP3A4KDM4EMAPTNPC1
SCHEMBL31470604 0.73 TDP1 (0.35) TDP1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL9505716 0.73 MAPT (0.38) TDP1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL27870146 0.73 ALDH1A1 (0.48) TDP1LMNACYP3A4IDO1KDM4E
SCHEMBL21594550 0.72 PTK2 (0.38) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3339305-A1 INDOLE DERIVATIVE, PREPARATION METHOD THEREOF, AND USE THEREOF IN PHARMACEUTICAL DRUG Zhejiang Hisun Pharmaceutical Co., Ltd (CN) 2018-06-27 EP disclosed